| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IDO1 |
3-Phenylpyridine |
NA |
161000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
Avicennol |
635000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(2-benzylphenyl)-2H-triazole |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1H-indazol-4-yl(trimethyl)silane |
NA |
NA |
150000 |
NA |
NA |
NA |
BindingDB |
| IDO1 |
4-[3-chloro-2-[(E)-2-cyclohexylethenyl]phenyl]-2H-triazole |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
N-(2-morpholin-4-ylethyl)-6-(4-phenylphenyl)imidazo[2,1-b][1,3]thiazol-5-amine |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
2-[[1-(2,4-Dichlorophenyl)-2-imidazol-1-ylethoxy]methyl]-1,3-benzoxazole |
NA |
136100 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
2-[[1-(2,4-Difluorophenyl)-2-imidazol-1-ylethoxy]methyl]-1,3-benzothiazole |
NA |
133100 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
4-Chloro-2-(3-methylimidazol-4-yl)aniline |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
2-(5-fluoro-1H-benzimidazol-2-yl)ethanamine |
NA |
NA |
548000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| IDO1 |
N-(azetidin-3-ylmethyl)-6-bromo-1H-indazol-4-amine |
NA |
112700 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
3-amino-4-[6-[bis(2-chloroethyl)amino]-1H-indol-3-yl]butanoic acid |
NA |
227000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
2-[(6-bromo-1H-indazol-4-yl)amino]-1-(4-hydroxyphenyl)ethanone |
NA |
137100 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
6-bromo-N-(pyrrolidin-3-ylmethyl)-1H-indazol-4-amine |
NA |
104900 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
(1S,2S)-2-[(6-bromo-1H-indazol-4-yl)methylamino]cyclohexan-1-ol |
NA |
203800 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
(1R,2S)-2-[[(5-chloro-1H-indazol-7-yl)amino]methyl]cyclohexan-1-ol |
NA |
178300 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
N-tert-butyl-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-5-amine |
NA |
281000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
6-pyridin-4-yl-N-(2,4,4-trimethylpentan-2-yl)imidazo[2,1-b][1,3]thiazol-5-amine |
NA |
691000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
3-[5-(2,4,4-Trimethylpentan-2-ylamino)imidazo[2,1-b][1,3]thiazol-6-yl]benzonitrile |
NA |
477000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
6-phenyl-N-(2,4,4-trimethylpentan-2-yl)imidazo[2,1-b][1,3]thiazol-5-amine |
NA |
465000 |
NA |
NA |
NA |
NA |
BindingDB |