| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IDO1 |
N-tert-butyl-6-pyridin-4-ylimidazo[2,1-b][1,3]thiazol-5-amine |
NA |
908000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
6-[4-(trifluoromethyl)phenyl]-N-(2,4,4-trimethylpentan-2-yl)imidazo[2,1-b][1,3]thiazol-5-amine |
NA |
1016000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
N-tert-butyl-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazol-5-amine |
NA |
1286000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
6-(1,3-benzodioxol-5-yl)-N-tert-butylimidazo[2,1-b][1,3]thiazol-5-amine |
NA |
1452000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
4-(Dimethylamino)naphthalen-1-ol |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-bromo-5-(4-methylphenyl)-2H-triazole |
NA |
1028000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1H-1,2,4-Triazole, 5-phenyl- |
NA |
580000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
Oxyquinoline |
NA |
750000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| IDO1 |
4-[4-(methylsulfanyl)phenyl]-1H-imidazole |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1-(3,4-dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol |
NA |
830000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1-[2-(2,4-Dichlorophenyl)ethyl]-1H-imidazole |
NA |
820000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(2-ethylphenyl)-2H-triazole |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
7,8-Dimethyl-10-(2-acetoxyethyl)isoalloxazine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
2-Amino-6-nitrobenzothiazole |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
5-(2-Fluorophenyl)-1H-imidazole |
NA |
179000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-(1H-1,2,3-Triazol-5-yl)benzaldehyde |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
3-(1H-imidazol-4-yl)phenol |
NA |
365000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(2,6-Dimethoxyphenyl)-1H-imidazole |
NA |
734000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1,2-bis(1H-benzimidazol-2-yl)ethane-1,2-diol |
NA |
NA |
774000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| IDO1 |
|
367000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |