Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| IDO1 | N-(2-(1,3-benzothiazol-2-ylthio)ethyl)aniline | NA | 115400 | NA | NA | NA | NA | BindingDB |
| IDO1 | ethyl 1-(4-chlorophenyl)-1H-1,2,3-triazole-4-carboxylate | NA | 2000000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 5-(1H-indol-3-ylmethyl)-3-methyl-2-thioxo-4-Imidazolidinone | NA | 115000 | NA | NA | NA | NA | BindingDB |
| IDO1 | 5h-Pyrido[3,4-b][1,4]benzothiazine | NA | 421600 | NA | NA | NA | NA | BindingDB |
| IDO1 | 1-Oxo-2-phenyl-1h-inden-3-yl acetate | NA | 266000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 1-[2-(1H-indol-3-yl)ethyl]-3-methylthiourea | 342300 | NA | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 2-(3-Bromoanilino)acetohydrazide | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| IDO1 | Benzophenone | NA | 1000000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| IDO1 | 1-(2,4-dichlorobenzyl)-1H-imidazole | NA | 310000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 2-(1H-imidazol-1-yl)aniline | NA | 1300000 | NA | NA | NA | NA | BindingDB |
| IDO1 | alpha-(2,4-Dichlorophenyl)-1H-imidazole-1-ethanol | NA | 130000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 2-(2-methylphenyl)-1H-phenanthro[9,10-d]imidazole | NA | 512000|464000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | Methyl 2-amino-2-(naphthalen-2-yl)acetate | NA | NA | 169000 | NA | NA | NA | BindingDB|ChEMBL |
| IDO1 | 1H-Benzo[a]carbazole-1,4(11H)-dione, 8-methoxy-11-methyl- | NA | 1000000 | NA | NA | NA | NA | TTD |
| IDO1 | Phenthiazamine | NA | 1000000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | Indoximod | NA | NA|1500000|2500000|696700|100000000 | NA | 110000|NA | NA | NA | BindingDB|PubChem|TTD |
| IDO1 | 2-(2-fluorophenyl)-1H-phenanthro[9,10-d]imidazole | NA | 231000|108000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | N-(2-(6-oxopyridazin-1(6H)-yl)ethyl)-2-naphthamide | NA | NA | 240000 | NA | NA | NA | BindingDB|ChEMBL |
| IDO1 | S-Hexyl-brassinin | 363600 | NA | NA | NA | NA | NA | TTD |
| IDO1 | N,N-dimethyl-1-(4-phenylthiazol-2-ylthio)methanamine | NA | 1000000 | NA | NA | NA | NA | TTD |