Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| IDO1 | 4-methyl-3-(2H-triazol-4-yl)aniline | NA | 3200000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | N-methyl-2-(2H-triazol-4-yl)aniline | NA | 1800000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 4-(4-chlorophenyl)-1H-1,2,3-triazole | NA | 530000|817000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 2-(3-chloro-2-fluorophenyl)isothiazol-3(2H)-one | NA | 200000 | NA | NA | NA | NA | BindingDB |
| IDO1 | Tryptophan | NA | 498700 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| IDO1 | 4-(4-bromophenyl)-1H-1,2,3-triazole | NA | 1256000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | Norharman | 180000 | NA | NA | NA | NA | NA | BindingDB |
| IDO1 | 4-(4-fluorophenyl)-1H-imidazole | NA | 123000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | N-[2-(5-phenylimidazol-1-yl)ethyl]acetamide | NA | 1000000 | NA | NA | NA | NA | TTD |
| IDO1 | 2-Hydroxy-1,4-naphthoquinone | NA | 675000 | NA | NA | NA | NA | PubChem|TTD |
| IDO1 | 1-methyl-L-tryptophan | NA | NA|118500|138500|380000|385000|498700 | NA | 120000|NA | NA | NA | BindingDB |
| IDO1 | Harmol | NA | 2000000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 5-[2-[2-(1H-imidazol-5-yl)phenoxy]ethyl]pyrimidine | NA | 154000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 2-(3-Methylimidazol-4-yl)aniline | NA | 1700000 | NA | NA | NA | NA | BindingDB |
| IDO1 | Stk727735 | NA | 195000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | 4(5)-Phenylimidazole | NA | 140000|143000|428000 | NA | NA | NA | NA | BindingDB |
| IDO1 | 2-Mercaptobenzothiazole | NA | 126000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| IDO1 | methyl (2E)-2-cyano-2-(2-oxo-1H-indol-3-ylidene)acetate | NA | 130000 | NA | NA | NA | NA | BindingDB |
| IDO1 | US10233190, Example 1389 | NA | 127000 | NA | NA | NA | NA | BindingDB|TTD |
| IDO1 | US10233190, Example 1370 | NA | 120000 | NA | NA | NA | NA | BindingDB |