| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IDO1 |
3-Hydroxy-2-naphthoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| IDO1 |
2-(1H-indol-1-yl)-N-(5-oxopyrrolidin-3-yl)acetamide |
NA |
NA |
237000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| IDO1 |
1H-Benzotriazole |
NA |
2570000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
Benzothiazole |
NA |
652000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| IDO1 |
Tryptanthrine |
NA |
498700 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
9-Hydroxyfluorene |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| IDO1 |
4-Aminodiphenylamine |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| IDO1 |
Benzenamine, 2-phenoxy- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
(5aR,6R)-2-fluoro-6-hydroxy-5a,6-dihydro-5H-indolo[2,1-b]quinazolin-12-one |
NA |
451000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(1,3-Dihydrophenanthro[9,10-d]imidazol-2-ylidene)cyclohexa-2,5-dien-1-one |
NA |
522000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-Chloroaniline |
NA |
1319000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
3-(1H-phenanthro[9,10-d]imidazol-2-yl)phenol |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
(E)-1-(benzofuran-3-yl)-3-morpholinoprop-2-en-1-one |
NA |
NA |
147000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| IDO1 |
4-Nitro-2,1,3-benzothiadiazole |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
3-Hydroxybenzophenone |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2,2'-Dithiobisbenzothiazole |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| IDO1 |
1-(1H-Indol-2-yl)-2-pyridin-3-yl-ethanone |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
2-(5H-imidazo[5,1-a]isoindol-5-yl)-1-piperidin-4-ylethanol;dihydrochloride |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
(10R)-14-hydroxy-10,13-dimethyl-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6,14-pentaene-12-thione |
NA |
174600 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
(10S)-6-chloro-14-hydroxy-10,13-dimethyl-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2(7),3,5,14-pentaene-12-thione |
NA |
119800 |
NA |
NA |
NA |
NA |
BindingDB |