| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IDO1 |
(10S)-4-chloro-14-hydroxy-10,13-dimethyl-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2(7),3,5,14-pentaene-12-thione |
NA |
113900 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
(10S)-6-bromo-14-hydroxy-10,13-dimethyl-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2(7),3,5,14-pentaene-12-thione |
NA |
109300 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
1H-Indazole |
NA |
NA |
360000 |
NA |
NA |
NA |
BindingDB |
| IDO1 |
1-Methyl-DL-tryptophan |
NA |
267000|328000|380000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
3-(1H-1,2,3-triazol-5-yl)phenol |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
3-(1H-1,2,3-triazol-4-yl)pyridine |
NA |
680000|708000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(4-fluorophenyl)-1H-1,2,3-triazole |
NA |
190000|580000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
5-(2-Methoxyphenyl)-1H-1,2,3-triazole |
NA |
1028000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazole |
NA |
2300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-Phenylindolone |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
5-(2-Bromophenyl)-1H-1,2,3-triazole |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
3-(2H-1,2,3-triazol-4-yl)aniline |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO2 |
N-(1,3-benzodioxol-5-yl)-2-{[5-(4-methylphenyl)[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]sulfanyl}acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| IDO2 |
Indoximod |
3300000|3900000|NA |
NA|148900|262750|262700 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| IGF1R |
2H-Indol-2-one, 3-(1,3-dihydro-3-oxo-2H-indol-2-ylidene)-1,3-dihydro- |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| IGF1R |
4-N-[(3-bromophenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IGF1R |
4-N-[(4-chlorophenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IGF1R |
4-N-[(4-methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IGF1R |
4-N-[(4-bromophenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IGF1R |
|
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB |