| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IKBKB |
1-ethyl-N-(3-hydroxypropyl)-2-oxo-2a,9-dihydrobenzo[cd]indole-6-sulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
3,4-dichloro-2-ethoxy-N-(2-hydroxypropyl)benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
1-ethyl-2-oxo-N-(3-sulfamoylphenyl)-2a,9-dihydrobenzo[cd]indole-6-sulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
2,5-diethoxy-N-[3-(1H-imidazol-1-yl)propyl]benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
2,5-diethoxy-N-[3-(1H-imidazol-1-yl)propyl]-4-methylbenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
Pyrrolopyridine, 9 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
7-methoxy-3,4,5,10-tetrahydro-1H-2,5-methanoazepino[3,4-b]indole-1-carboxylic Acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
6-Methoxy-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
1H-Pyrrolo(2,3-b)pyridine |
NA |
667000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKE |
(R)-2-((1-(1-hydroxycyclopropanecarbonyl)pyrrolidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
367000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
5-(4-((4-(4-(Oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-(1-oxa-6-azaspiro[3.4]octan-6-yl)benzonitrile |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
(R)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-(pyrrolidin-3-yloxy)benzonitrile |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
(R)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-(1-(tetrahydro-2H-pyran-4-yl)ethoxy)benzonitrile |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-Methoxy-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
215000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 267 |
NA |
264000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 159 |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
5-(4-((2,2-difluorobenzo[d][1,3]dioxol-5-yl)amino)-1,3,5-triazin-2-yl)-2-((tetrahydro-2H-pyran-4-yl)oxy)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
4-(2-cyano-4-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)phenoxy)-N-methylpiperidine-1-carboxamide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-((4-Methyl-1,2,3-thiadiazol-5-yl)methoxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
3-(4-((4-(4-(Oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |