| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IKBKE |
US10040781, Example 196 |
NA |
391000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 127 |
NA |
562000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 37 |
NA |
305000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 5 |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
N-(2-(4-(2-cyano-4-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)phenoxy)piperidin-1-yl)-2-oxoethyl)acetamide |
NA |
223000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 412 |
NA |
202000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-((3-(2-Hydroxyacetyl)-3-azabicyclo[3.1.1]heptan-6-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
676000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 548 |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 286 |
NA |
237000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)piperidin-4-yl)oxy)-5-(4-((5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 271 |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-((1-Methyl-2-oxohexahydropyrimidin-5-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 564 |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-(((3R,4S)-3-fluoro-1-(tetrahydrofuran-3-yl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
330000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 447 |
NA |
197000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-(((3R,4S)-3-fluoro-1-(oxetan-3-yl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
328000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
(R)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-((1-(oxetane-3-carbonyl)pyrrolidin-3-yl)oxy)benzonitrile |
NA |
197000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 126 |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 91 |
NA |
607000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 484 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |