| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IKBKE |
(S)-3-((1-(2-hydroxypropanoyl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 128 |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-((1-(2-Hydroxyacetyl)azetidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
5-(4-((2-methyl-4-morpholinophenyl)amino)-1,3,5-triazin-2-yl)-2-((tetrahydro-2H-pyran-4-yl)oxy)benzonitrile |
NA |
161000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 495 |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 381 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 593 |
NA |
660000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 600 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 597 |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 609 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 602 |
NA |
619000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 130 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 129 |
NA |
175000|619000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 598 |
NA |
720000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 608 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 335 |
NA |
834000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 606 |
NA |
494000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 601 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 596 |
NA |
403000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 594 |
NA |
232000 |
NA |
NA |
NA |
NA |
BindingDB |