| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IMPDH2 |
1-(3-Cyano-1-methyl-1H-indol-6-yl)-3-o-tolyl-urea |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
1-(3-Cyano-1H-indol-6-yl)-3-p-tolyl-urea |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
[(2S,3S,4R,5S)-5-(6-aminopurin-9-yl)-4-fluoro-3-hydroxyoxolan-2-yl]methoxy-[[[(2R,3S,4R,5S)-5-(3-carbamoylphenyl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methyl]phosphinic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
TTD |
| INMT |
3,4,5,7,8,9-hexahydro-2H-pyrrolo[1,2-a][1,3]diazepine |
NA |
852000 |
NA |
NA |
NA |
NA |
BindingDB |
| INMT |
5'-Methylthioadenosine |
700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| INMT |
2-Methyl-1,2-thiazol-3-imine;hydrochloride |
NA |
3283000 |
NA |
NA |
NA |
NA |
BindingDB |
| INPP5A |
[2,4-Bis(phosphonatomethyl)phenyl]methyl-dioxido-oxo-lambda5-phosphane |
148000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| INPP5A |
(1R,2R,4R)-Cyclohexane-1,2,4-tris (methlyenephosphate) |
144000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| INPP5A |
(1R,2R,4R)-Cyclohexane-1,2,4-tris (methylenephosphonate) |
535000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| INSR |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
NA |
622000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| INSR |
|
NA |
640000 |
NA |
NA |
NA |
NA |
BindingDB |
| INSR |
(Hydroxy-naphthalen-2-yl-methyl)-phosphonic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| INSR |
N-(2-aminophenyl)-4-[[4-(3-bromoanilino)quinazolin-6-yl]oxymethyl]benzamide |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| INSR |
Tyrphostin 47 |
NA |
640000 |
NA |
NA |
NA |
NA |
TTD |
| INSR |
[4-Amino-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-5-thiazolyl](2,3-dihydro-1,4-benzodioxin-6-yl)methanone |
NA |
71000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| INSR |
[4-Amino-2-[[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]amino]-5-thiazolyl](3-methoxyphenyl)methanone |
NA |
24000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| INSRR |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
NA |
182000 |
NA |
NA |
NA |
NA |
BindingDB |
| IP6K1 |
6-[(E)-2-pyridin-4-ylethenyl]-3H-quinazolin-4-one |
NA |
127000 |
NA |
NA |
NA |
NA |
BindingDB |
| IP6K1 |
3-methyl-6-[(E)-2-phenylethenyl]quinazolin-4-one |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB |
| IP6K1 |
6-[(E)-2-phenylethenyl]-3H-pyrido[2,3-d]pyrimidin-4-one |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |