| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IP6K1 |
8-amino-6-pyrrolidin-1-yl-3H-quinazolin-4-one |
NA |
189000 |
NA |
NA |
NA |
NA |
BindingDB |
| IP6K2 |
6-[(E)-2-phenylethenyl]-3H-quinazolin-4-one |
NA |
193000 |
NA |
NA |
NA |
NA |
BindingDB |
| IP6K3 |
6-pyrrolidin-1-yl-3H-quinazolin-4-one |
NA |
137000 |
NA |
NA |
NA |
NA |
BindingDB |
| IP6K3 |
6-[(E)-2-phenylethenyl]-3H-quinazolin-4-one |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB |
| IRAK1 |
6-(6-methoxyimidazo[1,2-a]pyridin-3-yl)-N-piperidin-4-ylpyridin-2-amine |
NA |
293000 |
NA |
NA |
NA |
NA |
TTD |
| IRAK1 |
N-(azetidin-3-yl)-6-(6-chloroimidazo[1,2-a]pyridin-3-yl)pyridin-2-amine |
NA |
195000 |
NA |
NA |
NA |
NA |
TTD |
| IRAK1 |
6-(6-chloroimidazo[1,2-a]pyridin-3-yl)-N-piperidin-3-ylpyridin-2-amine |
NA |
175000 |
NA |
NA |
NA |
NA |
TTD |
| IRAK1 |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| IRAK3 |
Pazopanib |
NA |
NA |
800000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
NA |
NA |
1900000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Mln8054 |
NA |
NA |
1400000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Gefitinib |
NA |
NA |
1500000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Canertinib |
NA |
NA |
3000000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
N-[(2R,3S,4S,6S)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N-methylbenzamide |
NA |
NA |
180000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Sns-032 |
NA |
NA |
2900000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Tandutinib |
NA |
NA |
730000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Sunitinib |
NA |
NA |
940000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Jnj-7706621 |
NA |
NA |
3400000 |
NA |
NA |
NA |
BindingDB |
| IRAK3 |
Tozasertib |
NA |
NA |
5600000 |
NA |
NA |
NA |
BindingDB |
| IRAK4 |
(1R,2S,3R,5R)-3-[[5-(1,3-benzothiazol-2-yl)-2-(cyclobutylamino)pyrimidin-4-yl]amino]-5-(hydroxymethyl)cyclopentane-1,2-diol |
NA |
403000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |