| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IKBKE |
US10040781, Example 610 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 603 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 599 |
NA |
176000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 123 |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
2-[[8-(2-Hydroxyacetyl)-8-azabicyclo[3.2.1]octan-3-yl]oxy]-5-[4-[4-[4-(oxetan-3-yl)piperazin-1-yl]anilino]-1,3-diaza-5-azoniacyclohexa-1,4,5-trien-2-yl]benzonitrile |
NA |
218000 |
NA |
NA |
NA |
NA |
BindingDB |
| IKBKE |
US10040781, Example 435 |
NA |
292000 |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH1 |
[(2S,3R,4S)-5-(2-chloro-6-oxo-1H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl dihydrogen phosphate |
120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH1 |
[(2S,3R,4S)-3,4-dihydroxy-5-(6-oxo-2-propyl-1H-purin-9-yl)oxolan-2-yl]methyl dihydrogen phosphate |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH1 |
[(2S,3R,4S)-3,4-dihydroxy-5-(2-methyl-6-oxo-1H-purin-9-yl)oxolan-2-yl]methyl dihydrogen phosphate |
600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH1 |
[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R)-5-(4-carbamoylfuran-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate |
135120 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH1 |
4-Hydroxy-2-methylacetophenone |
NA |
620000 |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH1 |
7-Chloro-4-aminoquinoline |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH2 |
[(2S,3R,4S)-3,4-dihydroxy-5-(2-methyl-6-oxo-1H-purin-9-yl)oxolan-2-yl]methyl dihydrogen phosphate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
[(2S,3R,4S)-3,4-dihydroxy-5-[6-oxo-2-(trifluoromethyl)-1H-purin-9-yl]oxolan-2-yl]methyl dihydrogen phosphate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
[(2S,3R,4S)-3,4-dihydroxy-5-[2-(hydroxymethyl)-6-oxo-1H-purin-9-yl]oxolan-2-yl]methyl dihydrogen phosphate |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
[(2S,3R,4S)-5-[2-(difluoromethyl)-6-oxo-1H-purin-9-yl]-3,4-dihydroxyoxolan-2-yl]methyl dihydrogen phosphate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
[(2S,3R,4S)-3,4-dihydroxy-5-[6-oxo-2-(2-phenylethyl)-1H-purin-9-yl]oxolan-2-yl]methyl dihydrogen phosphate |
NA |
460000 |
NA |
NA |
NA |
NA |
TTD |
| IMPDH2 |
[(2S,3S,4R)-5-(6-aminopurin-9-yl)-4-fluoro-3-hydroxyoxolan-2-yl]methoxy-[[[(2R,3S,4R)-5-(3-carbamoylphenyl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methyl]phosphinic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH2 |
|
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB |
| IMPDH2 |
|
NA |
460000 |
NA |
NA |
NA |
NA |
BindingDB |