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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ITGA2B Ac-Arg-Gly-Asn-Ser-NH2 NA 200000 NA NA NA NA TTD
ITGA2B Ac-Arg-Gly-Glu-Ser-NH2 NA 200000 NA NA NA NA TTD
ITGA2B Ac-Lys-Gly-Glu-Ser-NH2 NA 200000 NA NA NA NA TTD
ITGA2B 3-[4-amino(imino)methylamino-1-methylcarboxamido-(1S)-butylcarboxamidomethylcarboxamido]-3-[1-carbamoyl-2-(4-hydroxyphenyl)-(1S)-ethylcarbamoyl]propanoic acid NA 102000 NA NA NA NA TTD
ITGA2B Ac-Arg-Gly-Asp-Ser-NHEt NA 200000 NA NA NA NA TTD
ITGA2B cyclo(Arg-Gly-Asp-D-Pro-Pro-Gly) NA 200000 NA NA NA NA TTD
ITGA2B 4-(2-Bromoacetamido)-TEMPO 1000000 NA NA NA NA NA TTD
ITGA2B Cilengitide NA 244000|206000 NA NA NA NA PubChem
ITGA2B 3-{3-[(Piperidin-4-ylmethyl)-carbamoyl]-benzoylamino}-propionic acid NA 330000 NA NA NA NA TTD
ITGA2B 3-{[3-Oxo-2-(2-piperidin-4-yl-ethyl)-indane-5-carbonyl]-amino}-propionic acid NA 2300000 NA NA NA NA TTD
ITGA2B 2-[(4-Fluoro-2,6-dimethylbenzoyl)amino]-3-[4-[4-[(pyridin-2-ylamino)methyl]piperidin-1-yl]phenyl]propanoic acid NA 105000 NA NA NA NA TTD
ITGA2B [(S)-7-(6-Amino-pyridin-2-ylcarbamoyl)-4-methyl-3-oxo-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepin-2-yl]-acetic acid 160000 NA NA NA NA NA TTD
ITGA2B 3-{[6-(2-Piperidin-4-yl-ethylcarbamoyl)-pyridine-2-carbonyl]-amino}-propionic acid NA 300000 NA NA NA NA TTD
ITGA2B 1-[(2S)-2-[[4-[(diaminomethylideneamino)methyl]benzoyl]amino]propanoyl]piperidine-4-carboxylic acid NA 707945.78 NA NA NA NA TTD
ITGA2B 2-[1-[(2S)-2-[[4-(diaminomethylideneamino)benzoyl]amino]propanoyl]piperidin-4-yl]acetic acid NA 741310.24 NA NA NA NA TTD
ITGA2B 2-[1-[2-[[4-(Diaminomethylideneamino)benzoyl]-methylamino]acetyl]piperidin-4-yl]acetic acid NA 758577.58 NA NA NA NA TTD
ITGA2B 2-[1-[3-[[4-(Diaminomethylideneamino)benzoyl]amino]propanoyl]piperidin-4-yl]acetic acid NA 199526.23 NA NA NA NA TTD
ITGA2B 1-[(2S)-2-[(4-carbamimidoylbenzoyl)amino]propanoyl]piperidine-4-carboxylic acid NA 109647.82 NA NA NA NA TTD
ITGA2B 1-[3-[[4-(Diaminomethylideneamino)benzoyl]amino]propanoyl]piperidine-4-carboxylic acid NA 758577.58 NA NA NA NA TTD
ITGA2B Ac-Arg-Gly-D-Asp(1)-OH.N(1)Ser-NH2 NA 200000 NA NA NA NA TTD