| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGA2B |
1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-3-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]-3-methyl-2-oxopiperidine-3-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5S)-5-[[(3-amino-4-chlorobenzoyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5R)-5-[[(3-amino-4-chlorobenzoyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
16-Acetylamino-7-carbamoylmethyl-13-(3-guanidino-propyl)-3,3,14-trimethyl-6,9,12,15-tetraoxo-1,2-dithia-5,8,11,14-tetraaza-cycloheptadecane-4-carboxylic acid amide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
1-[4-[(5R)-5-[[(5-chlorothiophene-2-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
1-[4-[(5S)-5-[[(5-chlorothiophene-2-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
[16-Acetylamino-4-carbamoyl-13-(3-guanidino-propyl)-3,3,10-trimethyl-6,9,12,15-tetraoxo-1,2-dithia-5,8,11,14-tetraaza-cycloheptadec-7-yl]-acetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
[16-Acetylamino-4-carbamoyl-13-(4-guanidino-butyl)-3,3-dimethyl-6,9,12,15-tetraoxo-1,2-dithia-5,8,11,14-tetraaza-cycloheptadec-7-yl]-acetic acid |
NA |
385000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
16-(2-Acetylamino-6-amino-hexanoylamino)-7-carboxymethyl-3,3,13-trimethyl-6,9,12,15-tetraoxo-1,2-dithia-5,8,11,14-tetraaza-cycloheptadecane-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
H-Phe-Arg-Gly-Asp-OH |
NA |
947000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
(S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amino]-3-[4-(2,6-dichloro-benzyloxy)-phenyl]-propionic acid |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
H-Lys-Cys(1)-Asp-Pro-Cys(1)-OH |
NA |
250000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(S)-2-(4-Methoxy-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(4R,9R)-9-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2,10-dioxo-6,7-dithia-3,11-diaza-bicyclo[11.3.1]heptadeca-1(17),13,15-triene-4-carboxylic acid |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGA4 |
(4R,7S,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-10-methyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid |
NA |
182000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-methyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(4R,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGA4 |
(4R,11R)-11-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6,10-dioxo-1,2-dithia-5,9-diaza-cyclododecane-4-carboxylic acid |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGA4 |
H-D-Tyr-Cys(1)-Ser-Pro-Cys(1)-OH |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |