| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGA2B |
Ac-Arg-Ala-Asp-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
2-[(1R,6S,7R,8S,9R,23S,24R,25S)-19-[3-(diaminomethylideneamino)propyl]-7,8,24,25-tetrahydroxy-4,12,15,18,21-pentaoxo-26,27-dioxa-3,11,14,17,20-pentazatricyclo[21.2.1.16,9]heptacosan-13-yl]acetic acid |
NA |
198000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
(5S,8S)-3-[(S)-2-Carboxy-2-(2,4,6-trimethyl-benzenesulfonylamino)-ethylcarbamoyl]-8-(pyridin-2-ylaminomethyl)-1-oxa-2,7-diaza-spiro[4.4]non-2-ene-7-carboxylic acid benzyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
cyclo[D-Arg-Gly-D-Asp-Phe-Pro-D-Arg-Gly-D-Asp-Phe-Pro] |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
3-{[1-Oxo-9-phenyl-2-(2-piperidin-4-yl-ethyl)-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepine-8-carbonyl]-amino}-propionic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
3-(4-Piperazin-1-yl-benzoylamino)-propionic acid |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
Methyl 1-[2-[(4-carbamimidoylbenzoyl)-methylamino]acetyl]piperidine-4-carboxylate |
NA |
331131.12 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
(2S)-2-[(2-ethyl-4-fluoro-6-methylbenzoyl)amino]-3-[4-[4-[(pyridin-2-ylamino)methyl]piperidin-1-yl]phenyl]propanoic acid |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
(2R)-2-[(2-ethyl-4-fluoro-6-methylbenzoyl)amino]-3-[4-[4-[(pyridin-2-ylamino)methyl]piperidin-1-yl]phenyl]propanoic acid |
NA |
159000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
Ac-Arg-Gly-D-Asp-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 2-[benzyl-[(2R)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 2-[benzyl-[(2S)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 2-[benzyl-[(3R)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 2-[benzyl-[(3S)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-3-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-2-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]-2-oxopiperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]-3-methyl-2-oxopiperidine-3-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA2B |
ethyl 1-[4-[(5R)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |