| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGA4 |
H-Leu-Arg-Cys(1)-Asp-Pro-Cys(1)-OH |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(S)-2-{(S)-2-[(S)-2-((2S,3S)-2-Amino-3-methyl-pentanoylamino)-4-methyl-pentanoylamino]-3-carboxy-propionylamino}-3-methyl-butyric acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGA4 |
(3S,6R,11R,14S)-3-(hydroxymethyl)-6-[[4-(4-hydroxyphenyl)benzoyl]amino]-2,5,13-trioxo-8,9-dithia-1,4,12-triazabicyclo[12.3.0]heptadecane-11-carboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGA4 |
Glycyl-arginyl-glycyl-aspartyl-serine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
(S)-2-(3-Methoxy-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
[4-({[2-(Trifluoromethyl)phenyl]carbamoyl}amino)phenyl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
(S)-2-(2-Fluoro-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
117000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(S)-2-(4-Fluoro-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
121000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(S)-2-(3-Fluoro-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
176000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
N-(1-Carbamoyl-2-hydroxy-propyl)-3-{2-[(isoquinoline-3-carbonyl)-amino]-4-methyl-pentanoylamino}-succinamic acid |
NA |
465000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
cyclo[D-Ala-D-Pro-D-Phe-Leu-D-Asp-Thr] |
NA |
292000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
cyclo[D-Asp-D-Pro-D-His-Leu-D-Asp-Thr] |
NA |
301000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
cyclo[D-Asp-D-Pro-D-Phe-Leu-D-Asp-Thr] |
NA |
163000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
cyclo[D-Asp-D-Pro-D-Met-Leu-D-Asp-Thr] |
NA |
317000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
cyclo[D-Asp-D-Pro-D-Tyr-Leu-D-Asp-Thr] |
NA |
308000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(S)-3-((R)-5-Methyl-3-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-hexanoylamino)-3-phenyl-propionic acid |
NA |
262000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
[Benzyl-((S)-5-methyl-3-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-hexanoyl)-amino]-acetic acid |
NA |
247000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(E)-(R)-3-((R)-5-Methyl-3-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-hexanoylamino)-hex-4-enoic acid |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
Lithium;2-[[benzyl-[[2-[4-[(2-methylphenyl)carbamoylamino]phenyl]acetyl]amino]carbamoyl]amino]-3-methylbutanoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
(4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-cyclohexyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |