| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGA4 |
22-Amino-13-carbamoylmethyl-19-(3-guanidino-propyl)-10-(1-hydroxy-ethyl)-16-hydroxymethyl-7-isobutyl-6,9,12,15,18,21-hexaoxo-1,2-dithia-5,8,11,14,17,20-hexaaza-cyclotricosane-4-carboxylic acid amide |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(S)-2-[((R)-3-Acetyl-thiazolidine-4-carbonyl)-amino]-3-(4-hydroxy-phenyl)-propionic acid |
NA |
263000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
2-[(Adamantane-1-carbonyl)-amino]-3-{2-[(adamantane-1-carbonyl)-amino]-2-methoxycarbonyl-ethyldisulfanyl}-propionic acid methyl ester |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
2-[2-[3-[2-[2-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxopropyl]-4-[[2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]phenoxy]acetic acid |
NA |
169800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
2-[2-[3-(12-Aminododecylamino)-3-oxopropyl]-4-[[2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]phenoxy]acetic acid |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
N-(12-aminododecyl)-2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetamide |
NA |
151400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGA4 |
(3S)-4-[[(2S)-1-methoxy-3-methyl-1-oxobutan-2-yl]amino]-3-[[(2S)-4-methyl-2-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]pentanoyl]amino]-4-oxobutanoic acid |
NA |
703000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
3-[2-Hydroxy-5-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]phenyl]propanoic acid |
NA |
208900 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
3-[5-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-hydroxyphenyl]propanoic acid |
NA |
138000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
Benzyl 3-[5-[[2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]phenyl]propanoate |
NA |
102300 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
3-[2-[2-[(2-Methylpropan-2-yl)oxy]-2-oxoethoxy]-5-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]phenyl]propanoic acid |
NA |
151400 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
2-[4-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-[3-oxo-3-(2-phenylethylamino)propyl]phenoxy]acetic acid |
NA |
105900 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
3-[2-Hydroxy-4-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]phenyl]propanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
3-[4-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-hydroxyphenyl]propanoic acid |
NA |
146200 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
3-[4-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]phenyl]propanoic acid |
NA |
190100 |
NA |
NA |
NA |
NA |
TTD |
| ITGA4 |
Fibronectin CS1 Peptide |
NA |
824000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA5 |
3-[4-(6-Amino-hexyloxy)-phenyl]-2-(butane-1-sulfonylamino)-propionic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA5 |
3-[4-(7-Amino-heptyloxy)-phenyl]-2-benzyloxycarbonylamino-propionic acid |
NA |
450000 |
NA |
NA |
NA |
NA |
TTD |
| ITGA5 |
Arginyl-glycyl-aspartic acid |
NA |
830000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |