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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ITGA5 (S)-3-[2-((3-Methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-3-phenyl-propionic acid NA 500000 NA NA NA NA TTD
ITGA5 (S)-3-(4-Methoxy-phenyl)-3-[2-((3-methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-propionic acid NA 500000 NA NA NA NA TTD
ITGA5 (E)-(S)-3-[2-((3-Methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-hex-4-enoic acid NA 500000 NA NA NA NA TTD
ITGA5 (S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-propionic acid NA 500000 NA NA NA NA TTD
ITGA5 (S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amino]-3-[4-(2,6-dichloro-benzyloxy)-phenyl]-propionic acid NA 800000 NA NA NA NA TTD
ITGA5 H-Val-Thr-Gly-Arg-Gly-Asp-Ser-Pro-Ala-OH NA 1100000 NA NA NA NA BindingDB|TTD
ITGA5 3-[[2-[3-(4-carbamimidoylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]acetyl]amino]propanoic Acid NA 180000 NA NA NA NA BindingDB|TTD
ITGAL 1,4-Benzodioxan NA NA 10000000 NA NA NA BindingDB
ITGAL 1-Methylindole NA NA 1400000 NA NA NA BindingDB
ITGAL 2-Bromohippuric acid NA 313500 NA NA NA NA BindingDB
ITGAL Benzotript NA 169000 NA NA NA NA BindingDB
ITGAL (S)-2-(4-Fluoro-benzoylamino)-3-(1H-indol-3-yl)-propionic acid NA 136000 NA NA NA NA BindingDB
ITGAL (S)-2-(3-Chloro-benzoylamino)-3-(1H-indol-3-yl)-propionic acid NA 295000 NA NA NA NA BindingDB
ITGAL (2S,3S)-2-(2-Bromo-benzoylamino)-3-methyl-pentanoic acid NA 106000 NA NA NA NA BindingDB
ITGAL 2-Bromo-N-[(S)-1-hydroxycarbamoyl-2-(1H-indol-3-yl)-ethyl]-benzamide NA 140000 NA NA NA NA BindingDB
ITGAL (R)-2-(2-Bromo-benzoylamino)-3-naphthalen-2-yl-propionic acid NA 242500 NA NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-[(piperidine-1-carbonyl)-amino]-propionic acid NA 380000 NA NA NA NA BindingDB
ITGAL (S)-2-(3,5-Dichloro-benzoylamino)-3-(1H-indol-3-yl)-propionic acid NA 200000 NA NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-[(pyridine-3-carbonyl)-amino]-propionic acid NA 112000 NA NA NA NA BindingDB
ITGAL (S)-2-(3,4-Dichloro-benzoylamino)-3-(1H-indol-3-yl)-propionic acid NA 170500 NA NA NA NA BindingDB