| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGAV |
H-Gly-Gly-Gly-Gly-Arg-Gly-Asp-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly-Gly-Ser-OH |
NA |
1733000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
3-[(3S,6S,12S,38S,41S,44S)-6-(carboxymethyl)-12-[3-(diaminomethylideneamino)propyl]-38-[(1R)-1-hydroxyethyl]-3-(2-methylpropyl)-2,5,8,11,14,17,20,23,26,29,32,35,37,40,43-pentadecaoxo-1,4,7,10,13,16,19,22,25,28,31,34,36,39,42-pentadecazabicyclo[42.3.0]heptatetracontan-41-yl]propanoic acid |
NA |
522000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-Benzyloxycarbonylamino-3-[4-(3-tert-butylamino-2-hydroxy-propoxy)-phenyl]-propionic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[(6R,9S,12S,18S)-9-benzyl-6-carbamoyl-18-[3-(diaminomethylideneamino)propyl]-7-methyl-8,11,14,17,20-pentaoxo-2,7,10,13,16,19-hexazatricyclo[21.4.0.04,27]heptacosa-1(23),3,24,26-tetraen-12-yl]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[(2S,5S,8S,11S)-8-[4-(4-azidobutanoylamino)butyl]-5-benzyl-11-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid |
NA |
109600 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
4-Chlorophenylbiguanide |
NA |
148600 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-[2-(methylthio)phenyl]imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
1-(Diaminomethylidene)-2-(2,5-dichlorophenyl)guanidine |
NA |
100200 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-(2-ethoxyphenyl)imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
1-(2-Chlorophenyl)biguanide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-(5-chloro-2-methylphenyl)imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-(2-{2-hydroxy-4-[2-(4-methyl-4H-[1,2,4]triazol-3-ylsulfanyl)-acetylamino]-phenyl}-benzooxazol-6-yl)-2-(4-methyl-4H-[1,2,4]triazol-3-ylsulfaanyl)-acetamide |
NA |
162100 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-(4-(5-(4-Nitrophenoxy)-1,3-dioxoisoindolin-2-yl)benzamido)benzoic acid |
NA |
180400 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-{4-[(trifluoromethyl)thio]phenyl}imidodicarbonimidic diamide |
NA |
101400 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-[2-Chloro-5-(trifluoromethyl)phenyl]imidodicarbonimidic diamide |
NA |
127200 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[(1R,6S,7R,8S,9R,23S,24R,25S)-19-[3-(diaminomethylideneamino)propyl]-7,8,24,25-tetrahydroxy-4,12,15,18,21-pentaoxo-26,27-dioxa-3,11,14,17,20-pentazatricyclo[21.2.1.16,9]heptacosan-13-yl]acetic acid |
NA |
597000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
3-(3-(3-amino-N-propylpropanamido)-4-methyl-2-oxo-6-phenyl-5,6-dihydropyridin-1(2H)-yl)propanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
3-(3-(6-amino-N-propylhexanamido)-4-methyl-2-oxo-6-phenyl-5,6-dihydropyridin-1(2H)-yl)propanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
N-{6-(4-carbamimidoyl-phenyl)-1-[(S)-1-(4-methoxy-phenyl)-ethyl]-4-methyl-2-oxo-1,2,5,6-tetrahydro-pyridin-3-yl}-N-propyl-malonamic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
3-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-3-oxopropanoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |