| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB1 |
3-[4-(6-Amino-hexyloxy)-phenyl]-2-(butane-1-sulfonylamino)-propionic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[4-(7-Amino-heptyloxy)-phenyl]-2-benzyloxycarbonylamino-propionic acid |
NA |
450000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Arginyl-glycyl-aspartic acid |
NA |
830000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ITGB1 |
H-Lys-Cys(1)-Asp-Pro-Cys(1)-OH |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(4R,7S,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-10-methyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid |
NA |
182000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-methyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid |
NA |
350000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
H-D-Tyr-Cys(1)-Ser-Pro-Cys(1)-OH |
NA |
126000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
H-Leu-Arg-Cys(1)-Asp-Pro-Cys(1)-OH |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[5-(3-Guanidino-propylcarbamoyl)-2-oxo-1-aza-bicyclo[5.2.0]non-8-yl]-propionic acid |
NA |
1300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Ac-Asp-Arg-Leu-Asp-Ser-OH |
NA |
259000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Glycyl-arginyl-glycyl-aspartyl-serine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
[4-({[2-(Trifluoromethyl)phenyl]carbamoyl}amino)phenyl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Arginyl-glycyl-aspartyl-phenylalanine |
NA |
1546000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(R)-3-[(R)-5-(3-Guanidino-propylcarbamoyl)-2-oxo-1-aza-bicyclo[5.2.0]non-8-yl]-propionic acid |
NA |
3100000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
H-Vyavtgrgdspa-NH2 |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(S)-3-((R)-5-Methyl-3-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-hexanoylamino)-3-phenyl-propionic acid |
NA |
262000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
[Benzyl-((S)-5-methyl-3-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-hexanoyl)-amino]-acetic acid |
NA |
247000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(E)-(R)-3-((R)-5-Methyl-3-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-hexanoylamino)-hex-4-enoic acid |
NA |
103000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Lithium;2-[[benzyl-[[2-[4-[(2-methylphenyl)carbamoylamino]phenyl]acetyl]amino]carbamoyl]amino]-3-methylbutanoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(4R,7S,10R)-10-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-cyclohexyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
TTD |