| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB1 |
(S)-2-[((R)-3-Acetyl-thiazolidine-4-carbonyl)-amino]-3-(4-hydroxy-phenyl)-propionic acid |
NA |
263000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-[(Adamantane-1-carbonyl)-amino]-3-{2-[(adamantane-1-carbonyl)-amino]-2-methoxycarbonyl-ethyldisulfanyl}-propionic acid methyl ester |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-(3-(3-amino-N-propylpropanamido)-4-methyl-2-oxo-6-phenyl-5,6-dihydropyridin-1(2H)-yl)propanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-(3-(6-amino-N-propylhexanamido)-4-methyl-2-oxo-6-phenyl-5,6-dihydropyridin-1(2H)-yl)propanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-(((S)-6-(4-aminophenyl)-1-((S)-1-(4-methoxyphenyl)ethyl)-4-methyl-2-oxo-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-3-oxopropanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
N-{6-(4-carbamimidoyl-phenyl)-1-[(S)-1-(4-methoxy-phenyl)-ethyl]-4-methyl-2-oxo-1,2,5,6-tetrahydro-pyridin-3-yl}-N-propyl-malonamic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-3-oxopropanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
4-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)carbamoyl)-4-methoxy-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)carbamoyl)succinic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-({1-[(4-Aminophenyl)methyl]-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl}(propyl)carbamoyl)-4-methoxy-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-({1-[(4-Aminophenyl)methyl]-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl}(propyl)carbamoyl)butanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-[2-[3-[2-[2-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxopropyl]-4-[[2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]phenoxy]acetic acid |
NA |
169800 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-[2-[3-(12-Aminododecylamino)-3-oxopropyl]-4-[[2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]phenoxy]acetic acid |
NA |
123000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
N-(12-aminododecyl)-2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetamide |
NA |
151400 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Tirofiban |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ITGB1 |
(3S)-4-[[(2S)-1-methoxy-3-methyl-1-oxobutan-2-yl]amino]-3-[[(2S)-4-methyl-2-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]pentanoyl]amino]-4-oxobutanoic acid |
NA |
703000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[2-Hydroxy-5-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]phenyl]propanoic acid |
NA |
208900 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[5-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-hydroxyphenyl]propanoic acid |
NA |
138000 |
NA |
NA |
NA |
NA |
TTD |