| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB1 |
Benzyl 3-[5-[[2-[4-[(2,6-dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]phenyl]propanoate |
NA |
102300 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[2-[2-[(2-Methylpropan-2-yl)oxy]-2-oxoethoxy]-5-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]phenyl]propanoic acid |
NA |
151400 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
2-[4-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-[3-oxo-3-(2-phenylethylamino)propyl]phenoxy]acetic acid |
NA |
105900 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[2-Hydroxy-4-[[2-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]acetyl]amino]phenyl]propanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[4-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-hydroxyphenyl]propanoic acid |
NA |
146200 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[4-[[2-[4-[(2,6-Dimethylphenyl)carbamoylamino]phenyl]acetyl]amino]-2-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]phenyl]propanoic acid |
NA |
190100 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(S)-3-[2-((3-Methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-3-phenyl-propionic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(S)-3-(4-Methoxy-phenyl)-3-[2-((3-methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-propionic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(E)-(S)-3-[2-((3-Methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-hex-4-enoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(S)-3-(3,4-Dimethoxy-phenyl)-3-[2-((3-methoxy-propyl)-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetyl}-amino)-acetylamino]-propionic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
(S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amino]-3-[4-(2,6-dichloro-benzyloxy)-phenyl]-propionic acid |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
H-Val-Thr-Gly-Arg-Gly-Asp-Ser-Pro-Ala-OH |
NA |
1100000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
Fibronectin CS1 Peptide |
NA |
824000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB1 |
3-[[2-[3-(4-carbamimidoylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]acetyl]amino]propanoic Acid |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB2 |
Indole |
NA |
NA |
300000 |
NA |
NA |
NA |
PubChem |
| ITGB3 |
Arg-Gly-Asp-Arg-Gly-Asp |
NA |
619000|753000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
3-[4-(6-Amino-hexyloxy)-phenyl]-2-(butane-1-sulfonylamino)-propionic acid |
NA |
150000|330000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
2-(2,4-dichlorophenoxy)-N-(4-{[(2,6-dimethoxy-4-pyrimidinyl)amino]sulfonyl}phenyl)acetamide |
NA |
137000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
2-Benzyloxycarbonylamino-3-[4-(3-phenyl-propoxy)-phenyl]-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[5-[2-[[4-(1H-benzimidazol-2-ylamino)phenyl]methylamino]-2-oxoethyl]-6-oxo-11H-benzo[c][1]benzazepin-11-yl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |