| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB3 |
Ac-Arg-Gly-Asn-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ac-Arg-Gly-Glu-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ac-Lys-Gly-Glu-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-[4-amino(imino)methylamino-1-methylcarboxamido-(1S)-butylcarboxamidomethylcarboxamido]-3-[1-carbamoyl-2-(4-hydroxyphenyl)-(1S)-ethylcarbamoyl]propanoic acid |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ac-Arg-Gly-Asp-Ser-NHEt |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[(11R,14S,17S,23S)-14-benzyl-11-carbamoyl-23-[3-(diaminomethylideneamino)propyl]-13,16,19,22,25-pentaoxo-7,12,15,18,21,24-hexazatetracyclo[24.2.2.12,6.05,9]hentriaconta-1(29),2(31),3,5,8,26(30),27-heptaen-17-yl]acetic acid |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
2-[(6R,9S,12S,18S)-9-benzyl-6-carbamoyl-18-[3-(diaminomethylideneamino)propyl]-7-methyl-8,11,14,17,20-pentaoxo-2,7,10,13,16,19-hexazatricyclo[21.4.0.04,27]heptacosa-1(23),3,24,26-tetraen-12-yl]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
2-[(11R,14S,17S,23S)-14-benzyl-11-carbamoyl-23-[3-(diaminomethylideneamino)propyl]-12-methyl-13,16,19,22,25-pentaoxo-7,12,15,18,21,24-hexazatetracyclo[24.2.2.12,6.05,9]hentriaconta-1(29),2(31),3,5,8,26(30),27-heptaen-17-yl]acetic acid |
NA |
244000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
2-[(12R,15S,18S,24S)-15-benzyl-12-carbamoyl-24-[3-(diaminomethylideneamino)propyl]-13-methyl-14,17,20,23,26-pentaoxo-8,13,16,19,22,25-hexazatetracyclo[25.4.0.02,7.06,10]hentriaconta-1(31),2,4,6,9,27,29-heptaen-18-yl]acetic acid |
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
2-[(2S,5S,8S,11S)-8-[4-(4-azidobutanoylamino)butyl]-5-benzyl-11-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid |
NA |
109600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
cyclo(Arg-Gly-Asp-D-Pro-Pro-Gly) |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
4-(2-Bromoacetamido)-TEMPO |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
cyclo[Arg-Gly-Asp-Chg-gGlu(NH2)(NH2)] |
NA |
364000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
cyclo[Arg-Gly-Asp-Chg-N(Me)gGlu(NH2)(NH2)] |
NA |
1199000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
Cilengitide |
NA |
244000|206000 |
NA |
NA |
NA |
NA |
PubChem |
| ITGB3 |
3-{3-[(Piperidin-4-ylmethyl)-carbamoyl]-benzoylamino}-propionic acid |
NA |
330000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
4-Chlorophenylbiguanide |
NA |
148600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
3-{[3-Oxo-2-(2-piperidin-4-yl-ethyl)-indane-5-carbonyl]-amino}-propionic acid |
NA |
2300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
N-(2-(((5-Chloro-2-pyridinyl)amino)sulfonyl)phenyl)-4-(2-oxo-1(2H)-pyridinyl)benzamide |
NA |
136000|257000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
2-[(4-Fluoro-2,6-dimethylbenzoyl)amino]-3-[4-[4-[(pyridin-2-ylamino)methyl]piperidin-1-yl]phenyl]propanoic acid |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |