| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB3 |
(5S,8S)-3-[(S)-2-Carboxy-2-(2,4,6-trimethyl-benzenesulfonylamino)-ethylcarbamoyl]-8-(pyridin-2-ylaminomethyl)-1-oxa-2,7-diaza-spiro[4.4]non-2-ene-7-carboxylic acid benzyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
cyclo[D-Arg-Gly-D-Asp-Phe-Pro-D-Arg-Gly-D-Asp-Phe-Pro] |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-{[1-Oxo-9-phenyl-2-(2-piperidin-4-yl-ethyl)-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepine-8-carbonyl]-amino}-propionic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-(4-Piperazin-1-yl-benzoylamino)-propionic acid |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Methyl 1-[2-[(4-carbamimidoylbenzoyl)-methylamino]acetyl]piperidine-4-carboxylate |
NA |
331131.12 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-(3-(3-amino-N-propylpropanamido)-4-methyl-2-oxo-6-phenyl-5,6-dihydropyridin-1(2H)-yl)propanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-(3-(6-amino-N-propylhexanamido)-4-methyl-2-oxo-6-phenyl-5,6-dihydropyridin-1(2H)-yl)propanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
N-{6-(4-carbamimidoyl-phenyl)-1-[(S)-1-(4-methoxy-phenyl)-ethyl]-4-methyl-2-oxo-1,2,5,6-tetrahydro-pyridin-3-yl}-N-propyl-malonamic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-3-oxopropanoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
4-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)carbamoyl)-4-methoxy-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)carbamoyl)succinic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-({1-[(4-Aminophenyl)methyl]-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl}(propyl)carbamoyl)butanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
(S)-N-benzyl-3-{[(R)-1-(5-guanidino-pentanoyl)-pyrrolidine-2-carbonyl]-amino}-succinamic acid |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
N-[2-[1-[(5-chloropyridin-2-yl)amino]ethyl]phenyl]-4-(2-oxopyridin-1-yl)benzamide |
NA |
152000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
N-(4-chlorophenyl)-2-[[4-(2-oxopyridin-1-yl)benzoyl]amino]benzamide |
NA |
102000|171000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
1-[4-(Difluoromethylthio)phenyl]biguanide |
NA |
178100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
(2S)-2-[(2-ethyl-4-fluoro-6-methylbenzoyl)amino]-3-[4-[4-[(pyridin-2-ylamino)methyl]piperidin-1-yl]phenyl]propanoic acid |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
(2R)-2-[(2-ethyl-4-fluoro-6-methylbenzoyl)amino]-3-[4-[4-[(pyridin-2-ylamino)methyl]piperidin-1-yl]phenyl]propanoic acid |
NA |
159000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Phenyl Biguanide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |