| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB3 |
Tirofiban |
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| ITGB3 |
|
NA |
162100 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB3 |
N-[3-(methylthio)phenyl]imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ethyl 3-{[{[amino(imino)methyl]amino}(imino)methyl]amino}benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ac-Arg-Gly-D-Asp-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[benzyl-[(3S)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 2-[benzyl-[(2R)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 2-[benzyl-[(2S)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 2-[benzyl-[(3R)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 2-[benzyl-[(3S)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[benzyl-[(2R)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[benzyl-[(2S)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[benzyl-[(3R)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-3-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-2-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]-2-oxopiperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]-3-methyl-2-oxopiperidine-3-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
ethyl 1-[4-[(5R)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
1-[4-[(5S)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-3-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |