| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB5 |
N-(5-chloropyridin-2-yl)-2-[[4-(2-oxopyridin-1-yl)phenyl]sulfonylamino]benzamide |
NA |
1733000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB5 |
N-(4-chlorophenyl)-2-[[4-(2-oxopyridin-1-yl)benzoyl]amino]benzamide |
NA |
2945000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB5 |
N-(3-chlorophenyl)-2-[[4-(2-oxopyridin-1-yl)benzoyl]amino]benzamide |
NA |
522000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB6 |
Me-N(1)Arg-Gly-Asp-Chg-Glu(1)-NH2 |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB6 |
cyclo[Arg-Sar-Asp-Chg-gGlu(NH2)(NH2)] |
NA |
211000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITGB7 |
(S)-2-(4-Methoxy-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
122000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
(S)-2-(3-Methoxy-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
122000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
(S)-2-(2-Fluoro-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
(S)-2-(4-Fluoro-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
(S)-2-(3-Fluoro-benzylamino)-3-phenyl-propionic acid tert-butyl ester |
NA |
176000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
N-(1-Carbamoyl-2-hydroxy-propyl)-3-{2-[(isoquinoline-3-carbonyl)-amino]-4-methyl-pentanoylamino}-succinamic acid |
NA |
280000|465000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB7 |
cyclo[D-Ala-D-Pro-D-Phe-Leu-D-Asp-Thr] |
NA |
292000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
cyclo[D-Asp-D-Pro-D-His-Leu-D-Asp-Thr] |
NA |
301000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
cyclo[D-Asp-D-Pro-D-Phe-Leu-D-Asp-Thr] |
NA |
163000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
cyclo[D-Asp-D-Pro-D-Met-Leu-D-Asp-Thr] |
NA |
317000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
cyclo[D-Asp-D-Pro-D-Tyr-Leu-D-Asp-Thr] |
NA |
308000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
22-Amino-13-carbamoylmethyl-19-(3-guanidino-propyl)-10-(1-hydroxy-ethyl)-16-hydroxymethyl-7-isobutyl-6,9,12,15,18,21-hexaoxo-1,2-dithia-5,8,11,14,17,20-hexaaza-cyclotricosane-4-carboxylic acid amide |
NA |
175000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB7 |
2-[[(1R,4S,6R,7R,8S,10S)-1,10-dimethoxy-4-(2-methylpropoxymethyl)-7-phenylmethoxy-2,5,9-trioxatricyclo[8.4.0.03,8]tetradecan-6-yl]oxy]acetic acid |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITPKA |
6-N-benzyl-2-N-[(3-chlorophenyl)methyl]-7H-purine-2,6-diamine |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| ITPKA |
Purine, 7 |
NA |
138000 |
NA |
NA |
NA |
NA |
BindingDB |