| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGB3 |
N-[2-(methylthio)phenyl]imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
1-(Diaminomethylidene)-2-(2,5-dichlorophenyl)guanidine |
NA |
100200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
N-(2-ethoxyphenyl)imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
1-(2-Chlorophenyl)biguanide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
N-(5-chloro-2-methylphenyl)imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
N-(2-{2-hydroxy-4-[2-(4-methyl-4H-[1,2,4]triazol-3-ylsulfanyl)-acetylamino]-phenyl}-benzooxazol-6-yl)-2-(4-methyl-4H-[1,2,4]triazol-3-ylsulfaanyl)-acetamide |
NA |
162100 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-(4-(5-(4-Nitrophenoxy)-1,3-dioxoisoindolin-2-yl)benzamido)benzoic acid |
NA |
180400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
N-{4-[(trifluoromethyl)thio]phenyl}imidodicarbonimidic diamide |
NA |
101400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
N-[2-Chloro-5-(trifluoromethyl)phenyl]imidodicarbonimidic diamide |
NA |
127200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ITGB3 |
[(S)-7-(6-Amino-pyridin-2-ylcarbamoyl)-4-methyl-3-oxo-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepin-2-yl]-acetic acid |
160000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
3-{[6-(2-Piperidin-4-yl-ethylcarbamoyl)-pyridine-2-carbonyl]-amino}-propionic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
1-[(2S)-2-[[4-[(diaminomethylideneamino)methyl]benzoyl]amino]propanoyl]piperidine-4-carboxylic acid |
NA |
707945.78 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[1-[(2S)-2-[[4-(diaminomethylideneamino)benzoyl]amino]propanoyl]piperidin-4-yl]acetic acid |
NA |
741310.24 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[1-[2-[[4-(Diaminomethylideneamino)benzoyl]-methylamino]acetyl]piperidin-4-yl]acetic acid |
NA |
758577.58 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[1-[3-[[4-(Diaminomethylideneamino)benzoyl]amino]propanoyl]piperidin-4-yl]acetic acid |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
1-[(2S)-2-[(4-carbamimidoylbenzoyl)amino]propanoyl]piperidine-4-carboxylic acid |
NA |
109647.82 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
1-[3-[[4-(Diaminomethylideneamino)benzoyl]amino]propanoyl]piperidine-4-carboxylic acid |
NA |
758577.58 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ac-Arg-Gly-D-Asp(1)-OH.N(1)Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
Ac-Arg-Ala-Asp-Ser-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGB3 |
2-[(1R,6S,7R,8S,9R,23S,24R,25S)-19-[3-(diaminomethylideneamino)propyl]-7,8,24,25-tetrahydroxy-4,12,15,18,21-pentaoxo-26,27-dioxa-3,11,14,17,20-pentazatricyclo[21.2.1.16,9]heptacosan-13-yl]acetic acid |
NA |
597000|198000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |