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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
ITGB3
2-Benzyloxycarbonylamino-3-[4-(4-piperidin-4-yl-butoxy)-phenyl]-propionic acid
NA
158000
NA
NA
NA
NA
BindingDB
ITGB3
3-[4-(7-Amino-heptyloxy)-phenyl]-2-benzyloxycarbonylamino-propionic acid
NA
147000|315000
NA
NA
NA
NA
BindingDB|TTD
ITGB3
Arginyl-glycyl-aspartic acid
NA
130000|1000000
NA
NA
NA
NA
PubChem
ITGB3
3-{3-[(5-Carbamimidoyl-1H-indole-2-carbonyl)-amino]-butyrylamino}-3-phenyl-propionic acid
NA
125000
NA
NA
NA
NA
BindingDB|TTD
ITGB3
3-{2-[(5-Carbamimidoyl-1H-indole-2-carbonyl)-amino]-2-methyl-propionylamino}-3-phenyl-propionic acid
NA
250000
NA
NA
NA
NA
TTD
ITGB3
2-[5-[2-[[4-(1H-benzimidazol-2-ylamino)cyclohexyl]methylamino]-2-oxoethyl]-6-oxo-11H-benzo[c][1]benzazepin-11-yl]acetic acid
NA
1000000
NA
NA
NA
NA
TTD
ITGB3
{2-bromo-6-ethoxy-4-[(Z)-(8-methyl-3-oxo[1,3]thiazolo[3,2-a]benzimidazol-2(3H)-ylidene)methyl]phenoxy}acetic acid
NA
132000
NA
NA
NA
NA
BindingDB|TTD
ITGB3
m-Chlorophenylbiguanide
NA
190600
NA
NA
NA
NA
BindingDB|TTD
ITGB3
H-Gly-Arg-Gly-Asp-Arg-Gly-Asp-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly-Gly-Ser-OH
NA
152000
NA
NA
NA
NA
TTD
ITGB3
cyclo[Arg-Gly-Asp-Arg-Gly-Asp-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly]
NA
257000
NA
NA
NA
NA
TTD
ITGB3
H-Gly-Gly-Gly-Gly-Gly-Gly-Gly-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly-Gly-Ser-OH
NA
171000
NA
NA
NA
NA
TTD
ITGB3
2-Benzyloxycarbonylamino-3-[4-(3-tert-butylamino-2-hydroxy-propoxy)-phenyl]-propionic acid
NA
300000
NA
NA
NA
NA
TTD
ITGB3
Ac-D-Arg-Gly-Asp-Ser-NH2
NA
200000
NA
NA
NA
NA
TTD
ITGB3
Ac-Arg-Gly-Asp-D-Ser-NH2
NA
138000
NA
NA
NA
NA
TTD
ITGB3
Ac-Arg-Arg-Gly-Asp-Phe-NH2
NA
113000
NA
NA
NA
NA
TTD
ITGB3
Ac-Lys-Gly-Asp-Ser-NH2
NA
200000
NA
NA
NA
NA
TTD
ITGB3
Ac-Cit-Gly-Asp-Ser-NH2
NA
200000
NA
NA
NA
NA
TTD
ITGB3
Ac-His-Gly-Asp-Ser-NH2
NA
200000
NA
NA
NA
NA
TTD
ITGB3
Ac-Arg-Pro-Asp-Ser-NH2
NA
200000
NA
NA
NA
NA
TTD
ITGB3
Ac-Arg-Sar-Asp-Ser-NH2
NA
200000
NA
NA
NA
NA
TTD
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