| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ITGAV |
4-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)amino)-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)carbamoyl)-4-methoxy-4-oxobutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-((1-(4-Carbamimidoylbenzyl)-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl)(propyl)carbamoyl)succinic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-({1-[(4-Aminophenyl)methyl]-4-methyl-2-oxo-6-phenyl-1,2,5,6-tetrahydropyridin-3-yl}(propyl)carbamoyl)butanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
(S)-N-benzyl-3-{[(R)-1-(5-guanidino-pentanoyl)-pyrrolidine-2-carbonyl]-amino}-succinamic acid |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
1-[4-(Difluoromethylthio)phenyl]biguanide |
NA |
178100 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
Phenyl Biguanide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
Tirofiban |
NA |
260000 |
NA |
NA |
NA |
NA |
PubChem |
| ITGAV |
N-[3-(methylthio)phenyl]imidodicarbonimidic diamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
Ethyl 3-{[{[amino(imino)methyl]amino}(imino)methyl]amino}benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[benzyl-[(3S)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
ethyl 2-[benzyl-[(2R)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
ethyl 2-[benzyl-[(2S)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
ethyl 2-[benzyl-[(3R)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
ethyl 2-[benzyl-[(3S)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetate;2,2,2-trifluoroacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[benzyl-[(2R)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[benzyl-[(2S)-2-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
2-[benzyl-[(3R)-3-[(4-carbamimidoylphenoxy)methyl]-2,3-dihydro-1,4-benzodioxin-6-yl]amino]-2-oxoacetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
[1-((S)-4-Methyl-2-{2-[4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-pentanoyl)-piperidin-2-yl]-acetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ITGAV |
(S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amino]-3-[4-(2,6-dichloro-benzyloxy)-phenyl]-propionic acid |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |