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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ITGAL (S)-2-(3-Fluoro-benzoylamino)-3-(1H-indol-3-yl)-propionic acid NA 148000 NA NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-(2-methoxy-benzoylamino)-propionic acid NA 225000 NA NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-(3-methyl-benzoylamino)-propionic acid NA 295000 NA NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-(3-methoxy-benzoylamino)-propionic acid NA 438000 NA NA NA NA BindingDB
ITGAL 2,1,3-Benzothiadiazole NA NA 8000000 NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-(4-methoxy-benzoylamino)-propionic acid NA 178000 NA NA NA NA BindingDB
ITGAL (2R)-2-[(2-bromophenyl)formamido]-3-phenylpropanoicacid NA 280000 NA NA NA NA BindingDB
ITGAL N-Benzoyl-L-Tryptophan NA 127000 NA NA NA NA BindingDB
ITGAL (S)-3-(1H-Indol-3-yl)-2-(4-methyl-benzoylamino)-propionic acid NA 129000 NA NA NA NA BindingDB
ITGAL Indole NA NA 300000 NA NA NA BindingDB|PubChem
ITGAV Arg-Gly-Asp-Arg-Gly-Asp NA 546000 NA NA NA NA TTD
ITGAV 3-[4-(6-Amino-hexyloxy)-phenyl]-2-(butane-1-sulfonylamino)-propionic acid NA 330000 NA NA NA NA TTD
ITGAV 2-(2,4-dichlorophenoxy)-N-(4-{[(2,6-dimethoxy-4-pyrimidinyl)amino]sulfonyl}phenyl)acetamide NA 137000 NA NA NA NA TTD
ITGAV 3-[4-(7-Amino-heptyloxy)-phenyl]-2-benzyloxycarbonylamino-propionic acid NA 147000 NA NA NA NA TTD
ITGAV 3-{3-[(5-Carbamimidoyl-1H-indole-2-carbonyl)-amino]-butyrylamino}-3-phenyl-propionic acid NA 125000 NA NA NA NA TTD
ITGAV {2-bromo-6-ethoxy-4-[(Z)-(8-methyl-3-oxo[1,3]thiazolo[3,2-a]benzimidazol-2(3H)-ylidene)methyl]phenoxy}acetic acid NA 132000 NA NA NA NA TTD
ITGAV m-Chlorophenylbiguanide NA 190600 NA NA NA NA TTD
ITGAV H-Gly-Arg-Gly-Asp-Arg-Gly-Asp-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly-Gly-Ser-OH NA 152000 NA NA NA NA TTD
ITGAV cyclo[Arg-Gly-Asp-Arg-Gly-Asp-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly] NA 257000|380000 NA NA NA NA TTD
ITGAV H-Gly-Gly-Gly-Gly-Gly-Gly-Gly-Arg-Gly-Asp-Leu-Pro-Glu-Thr-Gly-Gly-Ser-OH NA 171000|2945000 NA NA NA NA TTD