| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IGF1R |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
NA |
NA |
210000 |
NA |
NA |
NA |
BindingDB |
| IGF1R |
N-(pyridin-3-ylmethyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| IGF1R |
Osimertinib |
NA |
2900000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| IGF1R |
AZ5104 |
NA |
263000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IGF1R |
N-(2-{2-Dimethylaminoethyl-methylamino}-4-methoxy-5-{[5-methyl-4-(1-methylindol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide |
NA |
196000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IGF1R |
[4-[(2S)-2-[[(2S)-2-acetamido-3-pyridin-3-ylpropanoyl]amino]-3-[[(2S)-1-[[(2S)-4-carboxy-1-[[(2S)-3-(4-chlorophenyl)-1-(methylamino)-1-oxopropan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-oxopropyl]benzoyl]-trihydroxyphosphanium |
NA |
489000 |
NA |
NA |
NA |
NA |
BindingDB |
| IGF1R |
[4-Amino-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-5-thiazolyl](2,3-dihydro-1,4-benzodioxin-6-yl)methanone |
NA |
22000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IGF1R |
[4-Amino-2-[[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]amino]-5-thiazolyl](3-methoxyphenyl)methanone |
NA |
20000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IGFBP5 |
(R)-2-((((9H-fluoren-9-yl)methoxy)carbonyl)amino)-3-(4-(tert-butoxy)phenyl)propanoic acid |
NA |
NA |
718000 |
NA |
NA |
NA |
BindingDB |
| IGFBP5 |
(2R)-2-(((9H-fluoren-9-ylmethoxy)carbonyl)amino)-4-methylpentanoic acid |
NA |
NA |
1088000 |
NA |
NA |
NA |
BindingDB |
| IGFBP5 |
Fmoc-D-Tyr(PO3H2)-OH |
NA |
NA |
1310000|1380000|1580000|1640000|1720000|1820000|1900000|2120000|2330000|2360000|2420000|2780000|2880000|2930000 |
NA |
NA |
NA |
BindingDB |
| IGFBP5 |
Dimethyl Sulfoxide |
NA |
NA |
541000000|610000000|648000000|650000000|719000000|783000000|921000000 |
NA |
NA |
NA |
BindingDB|PubChem |
| IGFBP5 |
(2R)-2-((((9H-fluoren-9-yl)methoxy)carbonyl)amino)-3-phenylpropanoic acid |
NA |
NA |
1075000 |
NA |
NA |
NA |
BindingDB |
| IKBKB |
2-(2-Quinolin-3-ylpyridin-4-YL)-1,5,6,7-tetrahydro-4H-pyrrolo(3,2-C)pyridin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
N-Phenyl-2-pyrimidinamine |
NA |
667000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
2-(2-(2-Fluorophenyl)pyridin-4-YL)-1,5,6,7-tetrahydro-4H-pyrrolo(3,2-C)pyridin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IKBKB |
4-[[4-(4-cyanophenyl)pyrimidin-2-yl]amino]-N-(2-hydroxyethyl)benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IKBKB |
4-[[4-(3-cyanophenyl)pyrimidin-2-yl]amino]-N-(2-hydroxyethyl)benzenesulfonamide |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IKBKB |
tert-butyl N-[2-[4-[2-(4-sulfamoylanilino)pyrimidin-4-yl]phenoxy]ethyl]carbamate |
NA |
138000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IKBKB |
3,4-dichloro-2-ethoxy-N-(1-hydroxybutan-2-yl)benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |