| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IDO1 |
(S)-2-amino-3-hydroxy-N-(4-hydroxynaphthalen-1-yl)propanamide |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-Amino-N-(4-hydroxynaphth-1-yl)acetamide |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
(S)-N-(4-hydroxynaphthalen-1-yl)pyrrolidine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
|
197000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
5-Iodo-4-phenyl-1H-1,2,3-triazole |
NA |
1371000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
8-Methylindolo[2,1-b]quinazoline-6,12-dione |
NA|218900 |
121200|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-Fluoroindolo[2,1-b]quinazoline-6,12-dione |
NA |
864400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1-(Carbamothioylamino)-3-(3,4-dichlorophenyl)urea |
NA |
NA |
941000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| IDO1 |
1-(1H-Indol-2-yl)-2-pyridin-3-yl-propan-1-one |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1-(4-Fluoro-1H-indol-2-yl)-2-pyridin-3-yl-ethanone |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1-(4,6-Dichloro-1H-indol-2-yl)-2-pyridin-3-yl-ethanone |
NA |
139000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
5-[2-(3-phenylpropoxy)phenyl]-1H-imidazole |
NA |
NA |
NA |
110000 |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-(5-Phenylimidazol-1-yl)ethanol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
N-methyl-2-(5-phenylimidazol-1-yl)acetamide |
NA |
187000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
5,6-Dihydroimidazo[1,5-d][1,4]benzoxazepine |
NA |
312000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
N-methyl-3-(5-phenylimidazol-1-yl)propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
4-(p-Tolyl)-1H-1,2,3-triazole |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(4-Methoxyphenyl)-1H-1,2,3-triazole |
NA |
6000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
3-methyl-2-(2H-triazol-4-yl)aniline |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2,2,2-trifluoro-N-[3-methyl-2-(2H-triazol-4-yl)phenyl]acetamide |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |