| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IDO1 |
5-[3-(Tert-butylamino)-7-methylimidazo[1,2-a]pyridin-2-yl]-2-methoxyphenol |
NA |
287000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
Brassinin derivative, 6 |
179600 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
Brassinin derivative, 14 |
363600 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
Brassinin derivative, 11 |
1267000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
Brassinin derivative, 10 |
149350 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(1H-indol-3-ylmethyl)-2-methyl-1,3-thiazole |
328700 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-[2-(trifluoromethyl)phenyl]-2H-triazole |
NA |
650000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
N-(1H-indol-3-ylmethyl)propanethioamide |
202000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
5-(4-Nitrophenyl)-4-nitro-1,2,3-triazole |
NA |
533000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(1H-Imidazol-4-yl)phenol |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
Methyl 3-aminonaphthalene-2-carboxylate |
NA |
460000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-[(2,4-dichlorophenyl)methylsulfanyl]-6-methyl-5H-pyrimidin-4-one |
NA |
217000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
1-(2-Chlorophenyl)-2-imidazol-1-ylethanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
2-(1H-tetrazol-5-yl)phenol |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
[4-(1,4-Dioxido-1,2,4-benzotriazin-3-yl)aminobutyl]-(2S)-N-tert-butoxycarbonyl-2-amino-(1-methyl-indole-3-yl)propanamide |
367000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
[5-(1,4-Dioxido-1,2,4-benzotriazin-3-yl)aminopentyl]-(2S)-N-tert-butoxycarbonyl-2-amino-(1-methyl-indole-3-yl)propanamide |
197000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
4-phenyl-1H-1,2,3-triazole |
NA |
143000|251200 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
(NE)-N-(2-phenyl-1,2-dihydroindol-3-ylidene)hydroxylamine |
NA |
510000|366000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
7-Fluoro-4-(2-fluoro-4-iodoanilino)-2,1,3-benzoxadiazole-5-carboxylic acid |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
4-[(2,4-dichlorophenyl)methylsulfanyl]-6-methyl-5,6-dihydro-1H-pyrimidin-2-one |
NA |
172000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |