| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HTR1A |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(2''-pyrimidyl)piperazine |
331000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(N-methyl)piperazine |
5000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(N-methyl)piperazine |
5000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(3,4-dihydroisoquinoline) |
1310000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-(3,4-dihydroisoquinoline) |
5000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) |
5000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) |
5000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2''-pyrimidyl)piperazine |
5000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3''-trifluoromethylphenyl)piperazine |
1308000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3''-trifluoromethyl)piperazine |
1409000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2''-methoxyphenyl)piperazine |
1092000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(4''-fluorophenyl)piperazine |
783000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
3-benzyl-2-phenyl-5-(pyridin-2-ylamino)-5-(trifluoromethyl)-3,5-dihydro-4H-imidazol-4-one |
284100 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR1A |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR1A |
8-(3,6-dihydro-2H-pyridin-1-yl)-3-thia-1,7-diazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene |
NA |
457088.19 |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
Pamidronic Acid |
NA |
NA |
NA |
NA |
NA |
113999 |
PubChem |
| HTR1A |
Pramoxine |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR1A |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR1A |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |