| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
(S)-5-(3-Fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide |
11152667 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
Regorafenib |
11167602 |
ChemBL, Pubchem |
| TTK |
HGNC:12401 |
P33981 |
4-{[(7r)-8-Cyclopentyl-7-Ethyl-5-Methyl-6-Oxo-5,6,7,8-Tetrahydropteridin-2-Yl]amino}-3-Methoxy-N-(1-Methylpiperidin-4-Yl)benzamide |
11364421 |
DSigDB, Pubchem |
| TTK |
HGNC:12401 |
P33981 |
Ast-487 |
11409972 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
Kw-2449 |
11427553 |
Pubchem |
| TTK |
HGNC:12401 |
P33981 |
N-(6-Oxo-1,6-Dihydro-3,4'-Bipyridin-5-Yl)benzamide |
11623444 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-(4-Methylpiperazin-1-Yl)-N-(2-Oxo-5-(Pyridin-4-Yl)-1,2-Dihydropyridin-3-Yl)benzamide |
11646783 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
FOSTAMATINIB |
11671467 |
DrugBank |
| TTK |
HGNC:12401 |
P33981 |
BX-912 |
11754511 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
Azd-1152hqpa |
16007391 |
ChemBL, Pubchem |
| TTK |
HGNC:12401 |
P33981 |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
16038120 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide |
16129448 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
Fedratinib |
16722836 |
Pubchem |
| TTK |
HGNC:12401 |
P33981 |
4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)-N-(4-(methylsulfonyl)phenyl)pyrimidin-2-amine |
16747683 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
Pictilisib |
17755052 |
Pubchem |
| TTK |
HGNC:12401 |
P33981 |
1-Methyl-8-[(2-methylphenyl)amino]-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide |
24992861 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[(9-Cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide |
25015677 |
GtoPDB |
| TTK |
HGNC:12401 |
P33981 |
Ruxolitinib |
25126798 |
Pubchem |
| TTK |
HGNC:12401 |
P33981 |
Omipalisib |
25167777 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
1-(4-(4-(2-(Isopropylsulfonyl)phenylamino)-1H-pyrrolo[2,3-b]pyridin-6-ylamino)-3-methoxyphenyl)piperidin-4-ol |
25195352 |
ChemBL, GtoPDB, TTD |