| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
5-fluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide |
25218614 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[[4-Amino-5-chloro-6-(2-propan-2-ylsulfonylanilino)-2-pyrimidinyl]amino]-3-methoxyphenyl]-4-piperidinecarboxamide |
25226117 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamide |
25226483 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
3-[(1R)-1-(2-chlorophenyl)ethoxy]-5-{6-[(1-methylpiperidin-4-yl)methoxy]-1H-1,3-benzodiazol-1-yl}thiophene-2-carboxamide |
25263124 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-2-(4-(4-Hydroxypiperidin-1-Yl)-2-Methoxyphenylamino)-5-Methyl-8,9-Dihydro-5h-Pyrimido[4,5-B][1,4]diazepin-6(7h)-One |
25271586 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
Foretinib |
42642645 |
Pubchem |
| TTK |
HGNC:12401 |
P33981 |
Pyrazolo[4,3-h]quinazoline-3-carboxamide, 1 |
44236351 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
Pyrazolo[4,3-h]quinazoline-3-carboxamide, 16 |
44236353 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[4-[4-(dimethylamino)piperidine-1-carbonyl]-2-methoxyanilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44555517 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[2-methoxy-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44555518 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[2-methoxy-4-[(2R)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44555519 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-(2-methoxyanilino)-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44555761 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[2-methoxy-4-(4-methyl-1,4-diazepane-1-carbonyl)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44555820 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
Nms-P715 |
44556162 |
ChemBL, GtoPDB, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44556163 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
8-[[4-(Aminocarbonyl)-2-methoxyphenyl]amino]-N-(2,6-diethylphenyl)-4,5-dihydro-1-methyl-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide |
44556214 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-8-[4-[2-(dimethylamino)ethylcarbamoyl]-2-methoxyanilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide |
44556329 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
WZ4002 |
44607530 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
Mps1-IN-2 |
44968267 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
4-[(9-cyclopentyl-5,8-dimethyl-6-oxo-7,8-dihydropyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidinyl)benzamide |
46843648 |
DSigDB |