| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-2-[[5-(4-hydroxypiperidin-1-yl)pyridin-2-yl]amino]-5-methyl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one |
46844026 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-2-[4-(4-hydroxy-4-methylpiperidin-1-yl)-2-methoxyanilino]-5-methyl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one |
46844085 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-2-[4-(4-hydroxypiperidin-1-yl)-2-propan-2-yloxyanilino]-5-methyl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one |
46844086 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-2-[2-ethoxy-4-(4-hydroxypiperidin-1-yl)anilino]-5-ethyl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one |
46844142 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-5-ethyl-2-[4-(4-hydroxypiperidin-1-yl)-2-propan-2-yloxyanilino]-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one |
46844143 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
9-Cyclopentyl-5-ethyl-2-[[5-(4-hydroxypiperidin-1-yl)pyridin-2-yl]amino]-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one |
46844145 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-[(2-Methoxyphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide |
46886960 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
Mpi-0479605 |
46909588 |
ChemBL, GtoPDB, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[[2-(2-methyl-4-morpholin-4-ylanilino)-7H-purin-6-yl]amino]cyclohexan-1-ol |
46927221 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
6-N-cyclohexyl-2-N-[4-morpholin-4-yl-2-(trifluoromethyl)phenyl]-7H-purine-2,6-diamine |
46927300 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
6-N-cyclohexyl-2-N-(2-ethoxy-4-morpholin-4-ylphenyl)-7H-purine-2,6-diamine |
46927301 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
6-cyclohexyloxy-N-(2-methyl-4-morpholin-4-ylphenyl)-7H-purin-2-amine |
46927371 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
2-N-(2-methyl-4-morpholin-4-ylphenyl)-6-N-(4-morpholin-4-ylcyclohexyl)-7H-purine-2,6-diamine |
46927447 |
TTD |
| TTK |
HGNC:12401 |
P33981 |
Torin 1 |
49836027 |
DSigDB |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-(8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazin-3-yl)benzamide |
50914591 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-(6-Bromo-8-(isobutylamino)imidazo[1,2-a]pyrazin-3-yl)-N-cyclopropylbenzamide |
50914592 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-(cyclopropylmethylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide |
50914874 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-Cyclopropyl-4-(8-isobutylamino-6-phenyl-imidazo[1,2-a]pyrazin-3-yl)-benzamide |
50914875 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(6-Oxo-1,6-Dihydro-3,4'-Bipyridin-5-Yl)-4-(Piperidin-1-Yl)benzamide |
52936434 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
1-methyl-8-(2-(trifluoromethoxy)phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide |
52947958 |
TTD |