| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-[cyclopropyl(thiophen-3-yl)methyl]-3-[4-(4-hydroxypiperidin-1-yl)phenyl]-1H-indazole-5-carboxamide |
89509755 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[cyclopropyl(phenyl)methyl]-3-[4-[1-[2-(dimethylamino)acetyl]piperidin-4-yl]oxyphenyl]-1H-indazole-5-carboxamide |
89509786 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
13-(4-bromo-2-methoxyanilino)-N,3-dimethyl-3,4,12,14-tetrazatricyclo[8.4.0.02,6]tetradeca-1(14),2(6),4,10,12-pentaene-5-carboxamide |
89895625 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[cyclopentyl(thiophen-3-yl)methyl]-3-[4-(1-methylpiperidin-4-yl)oxyphenyl]-1H-indazole-5-carboxamide |
89971805 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(cyclopentyl(pyridin-2-yl)methyl)-3-(4-((1-methylpiperidin-4-yl)oxy)phenyl)-1H-indazole-5-carboxamide |
89971850 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[4-(4-hydroxypiperidin-1-yl)phenyl]-1H-indazol-5-yl]-2-pyrrolidin-1-yl-2-thiophen-3-ylacetamide |
89971863 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[cyclopropyl(phenyl)methyl]-3-[4-[[(1S,5R)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]oxy]phenyl]-1H-indazole-5-carboxamide |
89971933 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2,3-Dihydroxypropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
89995566 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
6-[1-(2,2-difluoroethyl)pyrazol-4-yl]-N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]isoquinolin-3-amine |
89995571 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-6-(3-methyltriazol-4-yl)isoquinolin-3-amine |
89995587 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-6-(5-methylpyridin-3-yl)isoquinolin-3-amine |
89995589 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-(2-Chloro-4-morpholin-4-ylanilino)isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
89995623 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-6-[1-(oxan-4-ylmethyl)pyrazol-4-yl]isoquinolin-3-amine |
89995654 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[4-[3-[4-[3-(2-Hydroxy-2-methylpropyl)-2-methylimidazol-4-yl]-2-methoxyanilino]isoquinolin-6-yl]pyrazol-1-yl]-2-methylpropan-2-ol |
89995656 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[6-[1-(2-methoxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]phenyl]methanone |
89995733 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2-Hydroxy-3-methoxypropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
89995751 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2-Hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-[3-(methoxymethyl)azetidin-1-yl]methanone |
89995752 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-5-(1-methylpyrazol-4-yl)isoquinolin-3-amine |
89995972 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[5-(1-propan-2-ylpyrazol-4-yl)isoquinolin-3-yl]amino]phenyl]methanone |
89995973 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-6-methyl-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
89995975 |
ChemBL |