| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
8-(cyclohexylthio)-N-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidin-2-amine |
89995977 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2-(2-methoxyethoxy)-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-8-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995979 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2-ethoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-8-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995980 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
8-chloro-N-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidin-2-amine |
89995981 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[5-[1-(2-methoxyethyl)pyrazol-4-yl]isoquinolin-3-yl]amino]phenyl]methanone |
89995982 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[[[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]amino]methyl]cyclobutan-1-ol |
89995983 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(2-isopropoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-8-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995984 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
1-[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]azetidine-3-carbonitrile |
89995986 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(7-oxa-2-azaspiro[3.5]nonan-2-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995987 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(6-oxa-2-azaspiro[3.4]octan-2-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995988 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(2-oxa-7-azaspiro[4.4]nonan-7-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995989 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-6-methyl-8-(6-oxa-2-azaspiro[3.4]octan-2-yl)pyrido[3,4-d]pyrimidin-2-amine |
89995990 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-[1-(oxolan-3-yl)ethyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
89995994 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-[[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]amino]ethanol |
89995995 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[3-Methoxy-4-[[8-[(2-methoxy-2-methylpropyl)amino]pyrido[3,4-d]pyrimidin-2-yl]amino]phenyl]-2-methylpyrazol-3-yl]methanol |
89996000 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[8-[(2-methoxy-2-methylpropyl)amino]pyrido[3,4-d]pyrimidin-2-yl]amino]phenyl]methanone |
89996001 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[5-(3-methylimidazol-4-yl)isoquinolin-3-yl]amino]phenyl]methanone |
89996030 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(2,3-dimethylimidazol-4-yl)-2-methoxyphenyl]-5-(1-methylpyrazol-4-yl)-2,6-naphthyridin-3-amine |
89996035 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(2-ethoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-N8-(tetrahydro-2H-pyran-4-yl)pyrido[3,4-d]pyrimidine-2,8-diamine |
89996036 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-(oxetan-3-ylmethyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
89996037 |
ChemBL |