| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-[(3-methyloxetan-3-yl)methyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
89996042 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[4-(1,5-dimethylpyrazol-4-yl)-2-methoxyphenyl]-8-N-[(3-methyloxetan-3-yl)methyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
89996043 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[4-(1,5-dimethylpyrazol-4-yl)-2-methoxyphenyl]-8-(2-oxa-7-azaspiro[3.4]octan-7-yl)pyrido[3,4-d]pyrimidin-2-amine |
89996044 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-5-methyl-8-(6-oxa-2-azaspiro[3.4]octan-2-yl)pyrido[3,4-d]pyrimidin-2-amine |
89996046 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-5-methyl-8-N-[(3-methyloxolan-3-yl)methyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
89996047 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-(2-chloro-4-morpholin-4-ylphenyl)-8-N-(2,2-dimethylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
89996048 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-pyridin-4-ylpyrido[3,4-d]pyrimidin-2-amine |
89996049 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N8-cyclohexyl-N2-(4-(1-(2-(dimethylamino)ethyl)-1H-pyrazol-4-yl)-2-methoxyphenyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
89996101 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-(4-(3-methoxy-4-((8-((tetrahydro-2H-pyran-4-yl)amino)pyrido[3,4-d]pyrimidin-2-yl)amino)phenyl)-1H-pyrazol-1-yl)ethanol |
89996105 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(4-(1,2-dimethyl-1H-imidazol-5-yl)-2-methoxyphenyl)-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
89996108 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
3-[[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]amino]-2,2-dimethylpropan-1-ol |
89996117 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2,2-difluoropropyl)-2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
89996118 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-8-(pyrimidin-5-yl)pyrido[3,4-d]pyrimidin-2-amine |
89996120 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
1-[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]piperidine-4-carbonitrile |
89996123 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N8-cyclohexyl-N2-(2-methoxy-4-(1-(2-(4-methylpiperazin-1-yl)ethyl)-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
89996159 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N1-cyclohexyl-N7-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)-2,6-naphthyridine-1,7-diamine |
89996160 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-cyclopentyl-2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-methylpyrido[3,4-d]pyrimidine-2,8-diamine |
89996161 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(3,3-difluoropyrrolidin-1-yl)-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidin-2-amine |
89996162 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
6-cyclopropyl-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(2-oxa-7-azaspiro[3.4]octan-7-yl)pyrido[3,4-d]pyrimidin-2-amine |
89996163 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]morpholin-2-yl]methanol |
89996164 |
ChemBL |