| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TXK |
HGNC:12434 |
P42681 |
Crizotinib |
11626560 |
DSigDB, Pubchem |
| TXK |
HGNC:12434 |
P42681 |
FOSTAMATINIB |
11671467 |
DrugBank |
| TXK |
HGNC:12434 |
P42681 |
AZ-628 |
11676786 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
2,6-Dimethylphenyl (2,4-dimethoxyphenyl)(2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)carbamate |
11844351 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
R406 Benzenesulfonate |
11984591 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
16038120 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
Fedratinib |
16722836 |
Pubchem |
| TXK |
HGNC:12434 |
P42681 |
3-(4-Amino-7-piperidin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-phenol |
18792927 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
3-[[4-(5-Hydroxy-2-methylanilino)pyrimidin-2-yl]amino]benzenesulfonamide |
23657507 |
GtoPDB, TTD |
| TXK |
HGNC:12434 |
P42681 |
Benzamide, 3-[[4-[(5-methyl-1H-indazol-4-yl)amino]-2-pyrimidinyl]amino]- |
23657635 |
TTD |
| TXK |
HGNC:12434 |
P42681 |
Ibrutinib |
24821094 |
ChemBL, GtoPDB, Pubchem, TTD |
| TXK |
HGNC:12434 |
P42681 |
Ponatinib |
24826799 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
N-[1-(3-amino-3-oxopropyl)-5-[benzoyl(methyl)amino]benzimidazol-2-yl]-4-cyanobenzamide |
25110758 |
TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[1-(3-amino-3-oxopropyl)-5-[benzoyl(methyl)amino]benzimidazol-2-yl]-4-chlorobenzamide |
25110759 |
TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[5-(Benzoyl-ethyl-amino)-1-(2-carbamoyl-ethyl)-1H-benzoimidazol-2-yl]-4-cyano-benzamide |
25110760 |
TTD |
| TXK |
HGNC:12434 |
P42681 |
Lck inhibitor 2 |
25138012 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
3-({4-[(5-methyl-1H-indazol-4-yl)amino]pyrimidin-2-yl}amino)benzene-1-sulfonamide |
25138050 |
TTD |
| TXK |
HGNC:12434 |
P42681 |
2-Aminobenzimidazole with trans-stilbene, 8x |
25169253 |
TTD |
| TXK |
HGNC:12434 |
P42681 |
Foretinib |
42642645 |
Pubchem |
| TXK |
HGNC:12434 |
P42681 |
N-(1-(3-aminopropyl)-5-(N-methylcyclohexanecarboxamido)-1H-benzo[d]imidazol-2-yl)thiophene-2-carboxamide |
44432441 |
TTD |