| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TXK |
HGNC:12434 |
P42681 |
6-(trifluoromethyl)-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine |
44532526 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
(E)-N-(4-((4-Ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-(2-(4-methoxy-1H-pyrrolo[2,3-b]pyridin-5-yl)vinyl)-4-methylbenzamide |
53302361 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
4-Tert-Butyl-N-[2-Methyl-3-(6-{[4-(Morpholin-4-Ylcarbonyl)phenyl]amino}-7h-Purin-2-Yl)phenyl]benzamide |
53356518 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
Tirabrutinib |
54755438 |
ChemBL, Pubchem |
| TXK |
HGNC:12434 |
P42681 |
4-(2-fluorophenyl)-7-(4-methylpiperazine-1-carbonyl)-9H-carbazole-1-carboxamide |
56925034 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
4-(3-acetamido-2-methylphenyl)-7-(4-methylpiperazine-1-carbonyl)-9H-carbazole-1-carboxamide |
59375154 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
(2R)-2-(3-chloro-5-fluoroanilino)-2-cyclopropyl-N-[(3R)-1-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]acetamide |
67066715 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
(2R)-2-cyclopropyl-2-(3,5-dichloroanilino)-N-[(3R)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]acetamide |
67969590 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
2-(3,5-dichloroanilino)-N-[(3R)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]acetamide |
68064279 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
(2R)-2-cyclopropyl-2-(3,5-dichloroanilino)-N-[(3R)-1-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]acetamide |
68064412 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
7-(2-hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxoquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide |
70647728 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
4-[8-Azanyl-3-[(3~{r})-1-(3-Methyloxetan-3-Yl)carbonylpiperidin-3-Yl]imidazo[1,5-A]pyrazin-1-Yl]-~{n}-[4-(Trifluoromethyl)pyridin-2-Yl]benzamide |
71222614 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
(R)-4-(8-amino-3-(1-(3-methyloxetane-3-carbonyl)piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-3-fluoro-N-(4-(trifluoromethyl)-pyridin-2-yl)benzamide |
71226207 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
4-[8-Azanyl-3-[(3~{r},6~{s})-1-Cyclopropylcarbonyl-6-Methyl-Piperidin-3-Yl]imidazo[1,5-A]pyrazin-1-Yl]-3-Fluoranyl-~{n}-[4-(Trifluoromethyl)pyridin-2-Yl]benzamide |
71226367 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
Acalabrutinib |
71226662 |
ChemBL, GtoPDB, Pubchem |
| TXK |
HGNC:12434 |
P42681 |
US9718828, Example, 575 |
71226944 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
US9718828, Example, 551 |
71235465 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
Osimertinib |
71496458 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
Blk-IN-1 |
71519693 |
ChemBL, GtoPDB, TTD |
| TXK |
HGNC:12434 |
P42681 |
2-methyl-N-[2-({3-[2-(prop-2-enamido)acetamido]phenyl}amino)pyrimidin-5-yl]-5-[3-(trifluoromethyl)benzamido]benzamide |
71556703 |
ChemBL, GtoPDB, TTD |