| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TXK |
HGNC:12434 |
P42681 |
trans-4-[[4-[(6-Ethyl-2-benzothiazolyl)amino]-6-(phenylmethyl)-2-pyrimidinyl]amino]cyclohexanol |
73352604 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
Rilzabrutinib |
73388818 |
ChemBL, Pubchem |
| TXK |
HGNC:12434 |
P42681 |
(S,E)-2-(2-((4-amino-3-(2-fluoro-4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)pyrrolidine-1-carbonyl)-4-methyl-4-(methyl(oxetan-3-yl)amino)pent-2-enenitrile |
73389638 |
GtoPDB |
| TXK |
HGNC:12434 |
P42681 |
Atuzabrutinib |
73438222 |
ChemBL, Pubchem |
| TXK |
HGNC:12434 |
P42681 |
[2-methyl-5-[[3-(trifluoromethyl)phenyl]carbamoyl]phenyl] N-(2,4-dimethoxyphenyl)-N-[2-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]carbamate |
73707529 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
N-[2-methyl-5-[2-oxo-9-(1H-pyrazol-4-yl)-1-benzo[h][1,6]naphthyridinyl]phenyl]-2-propenamide |
73707530 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
4-(8-amino-3-((6R,8aS)-3-oxooctahydroindolizin-6-yl)imidazo[1,5-a]pyrazin-1-yl)-3-methoxy-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide |
76902376 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
4-(8-amino-3-((6R,8aS)-3-oxooctahydroindolizin-6-yl) imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide |
77105257 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
4-[3-[(6R,8aS)-1,1-dimethyl-3-oxo-6,7,8,8a-tetrahydro-5H-[1,3]oxazolo[3,4-a]pyridin-6-yl]-8-aminoimidazo[1,5-a]pyrazin-1-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide |
77106459 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
1-(2,4-Dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]urea |
78357808 |
DSigDB |
| TXK |
HGNC:12434 |
P42681 |
(Z)-2-[(2R)-2-[[4-amino-3-(2-fluoro-4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]pyrrolidine-1-carbonyl]-4-methyl-4-morpholin-4-ylpent-2-enenitrile |
86297191 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
Egfr-IN-1 |
86303858 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
10-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-[(2R)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl]amino]-6-oxopyridin-3-yl]pyridin-2-yl]-4,4-dimethyl-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-9-one |
86567260 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
3-chloro-4-(3-(5-chloro-1,3-dioxo-1H-pyrido[1,2-c]pyrimidin-2(3H)-yl)-2-methylphenyl)-7-(2-hydroxypropan-2-yl)-9H-carbazole-1-carboxamide |
86580694 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
Bms-986142 |
86582336 |
ChemBL, Pubchem, TTD |
| TXK |
HGNC:12434 |
P42681 |
Prn694 |
90044055 |
GtoPDB |
| TXK |
HGNC:12434 |
P42681 |
CID 90282962 |
90282962 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
4-[8-amino-3-[(6R,8aS)-3-oxo-2,5,6,7,8,8a-hexahydro-1H-indolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl]-3-cyclopropyloxy-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide |
90283326 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
Jak3-IN-1 |
92042864 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
Ritlecitinib |
118115473 |
ChemBL, Pubchem, TTD |