| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TXK |
HGNC:12434 |
P42681 |
N-(4-ethylpyridin-2-yl)-4-[6-(prop-2-enoylamino)quinolin-4-yl]oxybenzamide |
121273408 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
4-[6-(but-2-ynoylamino)-7-(2-morpholin-4-ylethoxy)quinolin-4-yl]oxy-N-pyridin-2-ylbenzamide |
121273567 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
2,3-dimethyl-4-[2-methyl-3-(prop-2-enoylamino)phenyl]-1H-indole-7-carboxamide |
121293882 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
Branebrutinib |
121293929 |
ChemBL, Pubchem |
| TXK |
HGNC:12434 |
P42681 |
4-[3-(ethenylsulfonylamino)-2-methylphenyl]-2,3-dimethyl-1H-indole-7-carboxamide |
121294143 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
4-[3-[[4-(dimethylamino)benzoyl]amino]-2-fluorophenyl]-7-(4-methylpiperazine-1-carbonyl)-9H-carbazole-1-carboxamide |
122191637 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[3-[[4-Amino-1-(4beta-hydroxycyclohexane-1alpha-yl)-1H-pyrazolo[3,4-d]pyrimidine-3-yl]ethynyl]-4-methylphenyl]-4-methyl-3-(trifluoromethyl)benzamide |
122419211 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
7-(2-methyl-4-phenoxyphenyl)-6-oxo-N-[(3R)-1-prop-2-enoylpyrrolidin-3-yl]-2-thia-5,7,11-triazatricyclo[6.3.1.04,12]dodeca-1(11),3,8(12),9-tetraene-3-carboxamide |
129219978 |
ChemBL |
| TXK |
HGNC:12434 |
P42681 |
US10266491, Example 10 |
132231876 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
5-(difluoromethyl)-N-[5-[[[(2S)-3,3-dimethylbutan-2-yl]amino]methyl]-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]thiophene-2-carboxamide |
134277578 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
5-(difluoromethyl)-N-[5-(morpholin-4-ylmethyl)-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]thiophene-2-carboxamide |
134277599 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
5-(2-oxo-1H-pyridin-4-yl)-N-[1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]thiophene-2-carboxamide |
134277617 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
4-cyano-N-[5-[[[(2S)-3,3-dimethylbutan-2-yl]amino]methyl]-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]benzamide |
134277633 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[5-[[[(2S)-3,3-dimethylbutan-2-yl]amino]methyl]-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]-5-(1,3-oxazol-5-yl)thiophene-2-carboxamide |
134277643 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
5-(2-aminopyridin-4-yl)-N-[1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]thiophene-2-carboxamide |
134277647 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[5-(methylamino)-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]-5-(1,3-oxazol-5-yl)thiophene-2-carboxamide |
134277652 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
5-[2-(methylamino)pyridin-4-yl]-N-[1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]thiophene-2-carboxamide |
134277654 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[5-[[[(2S)-3,3-dimethylbutan-2-yl]amino]methyl]-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]-1,3-thiazole-5-carboxamide |
134277685 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
N-[5-[[(4-hydroxycyclohexyl)amino]methyl]-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]-5-(1,3-oxazol-5-yl)thiophene-2-carboxamide |
134277696 |
ChemBL, TTD |
| TXK |
HGNC:12434 |
P42681 |
5-(difluoromethyl)-N-[5-[[(3-hydroxy-2,2-dimethylpropyl)amino]methyl]-1-(6-prop-2-enoyl-6-azaspiro[3.4]octan-2-yl)benzimidazol-2-yl]thiophene-2-carboxamide |
134277748 |
ChemBL, TTD |