GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
YES1 |
HGNC:12841 |
P07947 |
Momelotinib |
25062766 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Rebastinib |
25066467 |
ChemBL, DGidb, GtoPDB, Pubchem, TTD |
YES1 |
HGNC:12841 |
P07947 |
Cabozantinib s-malate |
25102846 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Cabozantinib |
25102847 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
Ruxolitinib |
25126798 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
Asp-3026 |
25134326 |
ChemBL, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
Lck inhibitor 2 |
25138012 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline |
25195294 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamide |
25226483 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
N-((1S)-2-(Dimethylamino)-1-phenylethyl)-6,6-dimethyl-3-((2-methylthieno(3,2-d)pyrimidin-4-yl)amino)-4,6-dihydropyrrolo(3,4-C)pyrazole-5(1H)-carboxamide |
25227462 |
ChemBL, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
3-[(2-chlorophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide |
25263092 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Vemurafenib |
42611257 |
DGidb, DSigDB |
YES1 |
HGNC:12841 |
P07947 |
Foretinib |
42642645 |
DGidb, DSigDB, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
Varlitinib |
42642648 |
ChemBL, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
7-(2,6-difluoro-4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)phenyl)-3-(1H-indazol-4-yl)-2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidine |
44187005 |
TTD |
YES1 |
HGNC:12841 |
P07947 |
(3Z)-N-methyl-3-[[3-(morpholin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-2-yl]methylidene]-2-oxo-1H-indole-5-sulfonamide |
44299176 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
(3Z)-5-ethylsulfonyl-3-[[3-(morpholin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-2-yl]methylidene]-1H-indol-2-one |
44299203 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
[4-(3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z)-ylidenemethyl]-4,5,6,7-tetrahydro-1H-indol-3-yl}-propyl)-piperazin-1-yl]-acetic acid |
44299236 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
5-Ethanesulfonyl-3-[1-{3-[3-(4-hydroxy-piperidin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one |
44299304 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
3-[1-{3-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide |
44299321 |
ChemBL, TTD |