GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
YES1 |
HGNC:12841 |
P07947 |
3-[1-{3-[3-(4-Methyl-piperazin-1-yl)-propyl]-4,5,6,7-tetrahydro-1H-indol-2-yl}-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide |
44299325 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
5-Ethanesulfonyl-3-[1-(3-{3-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-indol-2-yl)-meth-(Z)-ylidene]-1,3-dihydro-indol-2-one |
44299338 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
3-[2-[(Z)-(5-ethylsulfonyl-2-oxo-1H-indol-3-ylidene)methyl]-4,5,6,7-tetrahydro-1H-indol-3-yl]propanamide |
44299339 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
3-[1-(3-{3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-indol-2-yl)-meth-(Z)-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid methylamide |
44299354 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
(3Z)-N-methyl-3-[[3-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-indol-2-yl]methylidene]-2-oxo-1H-indole-5-sulfonamide |
44299360 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
[4-[2-acetamido-3-[[(1S)-1-[3-carbamoyl-4-(cyclohexylmethoxy)phenyl]ethyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
44313997 |
TTD |
YES1 |
HGNC:12841 |
P07947 |
SB-633825 |
44433173 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
(4-(7-(2-Chloro-5-hydroxyphenyl)-5-methylbenzo[e][1,2,4]triazin-3-ylamino)phenyl)(piperazin-1-yl)methanone |
44444041 |
TTD |
YES1 |
HGNC:12841 |
P07947 |
P505-15 |
44462758 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
Dabrafenib |
44462760 |
ChemBL, DSigDB, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
4-Methyl-3-[(7-pyridin-2-ylquinolin-4-yl)amino]phenol;hydrochloride |
44532204 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
N-(3-chloro-4-(3-fluorobenzyloxy)phenyl)-6-(5-((4-methylpiperazin-1-yl)methyl)furan-2-yl)thieno[3,2-d]pyrimidin-4-amine |
44571449 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
Sdccggsk-0000064.P001 |
44589696 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
7-(3-(azetidin-1-yl)cyclobutyl)-5-(3-(benzyloxy)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
45270897 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
Pha-793887 |
46191454 |
DGidb |
YES1 |
HGNC:12841 |
P07947 |
RN486 |
46908026 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
rac-2-(6-hydroxy-6-methylheptan-2-ylamino)-4-methyl-6-(5-methyl-1H-pyrazol-3-ylamino)nicotinonitrile hydrochloride |
46911726 |
TTD |
YES1 |
HGNC:12841 |
P07947 |
Gilteritinib |
49803313 |
ChemBL, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
Infigratinib |
53235510 |
TTD |
YES1 |
HGNC:12841 |
P07947 |
1-Tert-butyl-3-[7-(1-methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]urea |
53236670 |
ChemBL, TTD |