GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
YES1 |
HGNC:12841 |
P07947 |
N-[2-(dimethylamino)ethyl]-4-[[[1-(3-methoxyphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]hydrazinylidene]methyl]benzamide |
53239939 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
(E)-N-(4-((4-Ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-(2-(4-methoxy-1H-pyrrolo[2,3-b]pyridin-5-yl)vinyl)-4-methylbenzamide |
53302361 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
NG-25 |
53340664 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
7-methyl-5-(1-((3-(trifluoromethyl)phenyl)acetyl)-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo(2,3-d)pyrimidin-4-amine |
53469448 |
TTD |
YES1 |
HGNC:12841 |
P07947 |
5-Chloro-4-(1H-indol-3-yl)-N-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidin-2-amine |
56655374 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
Infigratinib Phosphate |
56669626 |
Pubchem |
YES1 |
HGNC:12841 |
P07947 |
2-phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine |
57332840 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-(4-morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-8-amine |
57332841 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
2-(4-methoxyphenyl)-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine |
57332844 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
2-(4-methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-8-amine |
57332969 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-(2,5-dimethoxyphenyl)-2-(4-methoxyphenyl)pyrido[3,4-b]pyrazin-8-amine |
57332970 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-phenyl-2-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine |
57332974 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
2-[4-[(4-Ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)anilino]-5,11-dimethyl-6-pyrimido[4,5-b][1,4]benzodiazepinone |
57340671 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
Spebrutinib |
59174488 |
GtoPDB |
YES1 |
HGNC:12841 |
P07947 |
4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-1-yl)-2-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine |
59757974 |
ChemBL, Pubchem |
YES1 |
HGNC:12841 |
P07947 |
5-[[7-(2,6-dimethylphenyl)-5-methyl-1,2,4-benzotriazin-3-yl]amino]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide |
59837608 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
2-[[7-(2,6-dimethylphenyl)-5-methyl-1,2,4-benzotriazin-3-yl]amino]-N-(2-pyrrolidin-1-ylethyl)-1,3-thiazole-4-carboxamide |
59837707 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
N-[4-(2-cyclopentylethoxy)phenyl]-7-(2,6-dimethylphenyl)-5-methyl-1,2,4-benzotriazin-3-amine |
59837783 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
N-[3-(diethylaminomethoxy)phenyl]-7-(2,6-dimethylphenyl)-5-methyl-1,2,4-benzotriazin-3-amine |
59837796 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
2,6-difluoro-N-[3-fluoro-4-[6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinolin-4-yl]oxyphenyl]benzenesulfonamide |
67073846 |
ChemBL |