GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ACHE |
N-[chloro-(4-methylphenoxy)phosphoryl]-N-methylmethanamine |
NA |
1370000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
2-Butylsulfanylcarbonyloxyethyl(trimethyl)azanium;chloride |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
(2-Butylsulfanylcarbonyloxy-ethyl)-trimethyl-ammonium; chloride |
NA |
500000|1000000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
3-(2-Morpholinoethylamino)-4-trifluoromethyl-6-phenylpyridazine |
NA |
740000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
2-(4-Ethylphenyl)sulfanylcarbonyloxyethyl-trimethylazanium;chloride |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
[2-(4-Ethyl-phenylsulfanylcarbonyloxy)-ethyl]-trimethyl-ammonium; chloride |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
Trimethyl(2-phenylsulfanylcarbonyloxyethyl)azanium;chloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Trimethyl-(2-phenylsulfanylcarbonyloxy-ethyl)-ammonium; chloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
N'-benzyl-N'-methyl-N-(6-phenylpyridazin-3-yl)ethane-1,2-diamine |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
16-Methoxy-11-methyl-3,5-dioxa-11-azapentacyclo[10.7.1.02,6.08,20.014,19]icosa-1(19),2(6),7,12(20),13,16-hexaene-15,18-dione |
NA |
221100 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
2-Ethylsulfanylcarbonyloxyethyl(trimethyl)azanium;chloride |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Trimethyl(2-propylsulfanylcarbonyloxyethyl)azanium;chloride |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
(3-Morpholin-4-ylpropyl)(6-phenylpyridazin-3-yl)amine |
NA |
410000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Deguelin |
NA |
126700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
9-Amino-2,3-dimethyl-2,3-dihydro-1H-cyclopenta[b]quinolin-3-ol |
NA |
134000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
9-[4-[(4-Fluorophenyl)methoxy]-3-methoxyphenyl]-2,3,4,5,6,7,9,10-octahydroacridine-1,8-dione |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
N-[fluoro-(4-methylphenoxy)phosphoryl]-N-methylmethanamine |
NA |
4290000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
Trimethyl-[2-(2-methylbutylsulfanylcarbonyloxy)ethyl]azanium;chloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Trimethyl-[2-(2-methyl-butylsulfanylcarbonyloxy)-ethyl]-ammonium; chloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
3-[methyl(prop-2-yn-1-yl)amino]-2,3-dihydro-1H-inden-4-yl N,N-dimethylcarbamate |
NA |
730000 |
NA |
NA |
NA |
NA |
BindingDB |