GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ACHE |
Flaxedil |
NA |
2110000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
3-(3,4-dimethoxyphenyl)-8,8-dimethyl-4H,8H-pyrano[2,3-f]chromen-4-one |
NA |
131170 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Ibuprofen |
NA |
235000|235110 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
ACHE |
2-(Trimethylammonium)ethyl thiol |
NA |
439541.62 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
N-(dimorpholin-4-ylphosphoryl)benzamide |
NA |
4150000 |
2954000 |
NA |
NA |
NA |
BindingDB |
ACHE |
[(Ethylimino)dimethanediyl]bis(phosphonic acid) |
NA |
22090000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
8,20-Diazatetracyclo[10.8.0.0^{2,7}.0^{14,19}]icosa-1(12),2(7),3,5,13,15,17,19-octaen-13-amine |
NA |
391100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
6,7-Dihydro-5h-benzo[6,7]cyclohepta[1,2-b]quinolin-8-amine |
NA |
166100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
6-Hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid |
NA |
186400|3995000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
(3-Methoxy-phenyl)-trimethyl-ammonium |
NA |
597035.29 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
1-(5-Pyridin-1-ium-1-ylpentyl)pyridin-1-ium |
NA |
1270000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
(3,4-Dimethoxyphenyl)-(4-morpholin-4-ylmethylphenyl)methanone |
NA |
345000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Clorgyline |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
2-(4-Hydroxy-3-methoxyphenyl)-2-pyrrolidin-1-ylacetonitrile |
NA |
358200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
2-(3-Hydroxy-4-methoxyphenyl)-2-pyrrolidin-1-ylacetonitrile |
NA |
394000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
2-(3-Hydroxy-4-methoxyphenyl)-2-piperidin-1-ylacetonitrile |
NA |
478000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
2-(3-Hydroxy-4-methoxyphenyl)-2-morpholin-4-ylacetonitrile |
NA |
363000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
(5-Bromo-pentyl)-trimethyl-ammonium |
NA |
534564.36 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Naringenin |
NA |
2045000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
ACHE |
(S)-Scoulerine |
NA |
143300 |
NA |
NA |
NA |
NA |
BindingDB |