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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC29A1 Adenosine, N-[(3-methoxyphenyl)methyl]- NA 114815.36 NA NA NA NA BindingDB|TTD
SLC29A1 Imipenem NA NA NA NA NA 300000 PubChem
SLC29A1 n6-2-Propyl adenosine NA 257039.58 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3R,4S,5R)-2-[2-amino-6-(3-methyl-5-nitroimidazol-4-yl)sulfanylpurin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol NA 575439.94 NA NA NA NA BindingDB|TTD
SLC29A1 (1R,3S,4R,5S)-1-(6-aminopurin-9-yl)-4-(hydroxymethyl)bicyclo[3.1.0]hexan-3-ol NA 626000 NA NA NA NA BindingDB
SLC29A1 (2R,3R,4S,5R)-2-(2-amino-6-methylsulfanylpurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol NA 204173.79 NA NA NA NA BindingDB|TTD
SLC29A1 6-Methylsulfanyl-9-(oxan-2-yl)purine NA 275422.87 NA NA NA NA BindingDB|TTD
SLC29A1 9H-Purin-2-amine, 9-butyl-6-(methylthio)- NA 218776.16 NA NA NA NA BindingDB|TTD
SLC29A1 6-Propan-2-ylsulfanyl-9-propylpurin-2-amine NA 144543.98 NA NA NA NA BindingDB|TTD
SLC29A1 9-Butyl-6-propan-2-ylsulfanylpurin-2-amine NA 120226.44 NA NA NA NA BindingDB|TTD
SLC29A1 1-(2-((2S,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yloxy)-4,6-dihydroxyphenyl)-3-(4-hydroxyphenyl)propan-1-one 1000000 NA NA NA NA NA TTD
SLC29A1 7H-Pyrrolo[2,3-d]pyrimidine-4-thiol, 7-beta-D-ribofuranosyl- NA 389045.14 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-[4-(1-piperidyl)pyrrolo[2,3-d]pyrimidin-7-yl]tetrahydrofuran-3,4-diol NA 194984.46 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-(4-methoxypyrrolo[2,3-d]pyrimidin-7-yl)tetrahydrofuran-3,4-diol NA 338844.16 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3R,4S,5R)-2-(5-bromo-4-methylsulfanyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol NA 114815.36 NA NA NA NA BindingDB|TTD
SLC29A1 Cefazolin NA NA NA NA NA 300000 PubChem
SLC29A1 N-(3-methylbutyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine NA 234422.88 NA NA NA NA BindingDB|TTD
SLC29A1 Meropenem NA NA NA NA NA 300000 PubChem
SLC29A1 (1R,13R,14S,15R)-7-(8-nitro-3,4-dihydro-1H-isoquinolin-2-yl)-11,16-dioxa-2,4,6,9-tetrazatetracyclo[11.2.1.02,10.03,8]hexadeca-3(8),4,6,9-tetraene-14,15-diol NA 1737800 NA NA NA NA BindingDB
SLC29A1 (1R,13R,14S,15R)-7-(5-nitro-3,4-dihydro-1H-isoquinolin-2-yl)-11,16-dioxa-2,4,6,9-tetrazatetracyclo[11.2.1.02,10.03,8]hexadeca-3(8),4,6,9-tetraene-14,15-diol NA 7413102.41 NA NA NA NA BindingDB