GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC29A1 |
Adenosine, N-[(3-methoxyphenyl)methyl]- |
NA |
114815.36 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC29A1 |
n6-2-Propyl adenosine |
NA |
257039.58 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3R,4S,5R)-2-[2-amino-6-(3-methyl-5-nitroimidazol-4-yl)sulfanylpurin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
575439.94 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(1R,3S,4R,5S)-1-(6-aminopurin-9-yl)-4-(hydroxymethyl)bicyclo[3.1.0]hexan-3-ol |
NA |
626000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC29A1 |
(2R,3R,4S,5R)-2-(2-amino-6-methylsulfanylpurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
204173.79 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
6-Methylsulfanyl-9-(oxan-2-yl)purine |
NA |
275422.87 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
9H-Purin-2-amine, 9-butyl-6-(methylthio)- |
NA |
218776.16 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
6-Propan-2-ylsulfanyl-9-propylpurin-2-amine |
NA |
144543.98 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
9-Butyl-6-propan-2-ylsulfanylpurin-2-amine |
NA |
120226.44 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
1-(2-((2S,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yloxy)-4,6-dihydroxyphenyl)-3-(4-hydroxyphenyl)propan-1-one |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC29A1 |
7H-Pyrrolo[2,3-d]pyrimidine-4-thiol, 7-beta-D-ribofuranosyl- |
NA |
389045.14 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-[4-(1-piperidyl)pyrrolo[2,3-d]pyrimidin-7-yl]tetrahydrofuran-3,4-diol |
NA |
194984.46 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-(4-methoxypyrrolo[2,3-d]pyrimidin-7-yl)tetrahydrofuran-3,4-diol |
NA |
338844.16 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3R,4S,5R)-2-(5-bromo-4-methylsulfanyl-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol |
NA |
114815.36 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC29A1 |
N-(3-methylbutyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
NA |
234422.88 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC29A1 |
(1R,13R,14S,15R)-7-(8-nitro-3,4-dihydro-1H-isoquinolin-2-yl)-11,16-dioxa-2,4,6,9-tetrazatetracyclo[11.2.1.02,10.03,8]hexadeca-3(8),4,6,9-tetraene-14,15-diol |
NA |
1737800 |
NA |
NA |
NA |
NA |
BindingDB |
SLC29A1 |
(1R,13R,14S,15R)-7-(5-nitro-3,4-dihydro-1H-isoquinolin-2-yl)-11,16-dioxa-2,4,6,9-tetrazatetracyclo[11.2.1.02,10.03,8]hexadeca-3(8),4,6,9-tetraene-14,15-diol |
NA |
7413102.41 |
NA |
NA |
NA |
NA |
BindingDB |